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Details

Stereochemistry RACEMIC
Molecular Formula C23H35N3O
Molecular Weight 369.5435
Optical Activity ( + / - )
Defined Stereocenters 2 / 2
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of ACTISOMIDE

SMILES

CC(C)N(CC[C@]1([C@H]2CCCCN2C(C)=NC1=O)C3=CC=CC=C3)C(C)C

InChI

InChIKey=QAHRRCMLXFLZTF-FYYLOGMGSA-N
InChI=1S/C23H35N3O/c1-17(2)25(18(3)4)16-14-23(20-11-7-6-8-12-20)21-13-9-10-15-26(21)19(5)24-22(23)27/h6-8,11-12,17-18,21H,9-10,13-16H2,1-5H3/t21-,23-/m1/s1

HIDE SMILES / InChI

Molecular Formula C23H35N3O
Molecular Weight 369.5435
Charge 0
Count
MOL RATIO 1 MOL RATIO (average)
Stereochemistry ABSOLUTE
Additional Stereochemistry No
Defined Stereocenters 2 / 2
E/Z Centers 0
Optical Activity UNSPECIFIED

Description

ACTISOMIDE is a class 1A/1B antiarrhythmic agent. It blocks sodium channels in a manner similar to lidocaine and mexiletine. It is a well-tolerated, effective agent against both atrial and ventricular arrhythmias.

Approval Year

PubMed

Substance Class Chemical
Record UNII
IJQ29N87NR
Record Status Validated (UNII)
Record Version