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Details

Stereochemistry ABSOLUTE
Molecular Formula C21H24F3N3O4.CH4O3S
Molecular Weight 535.534
Optical Activity UNSPECIFIED
Defined Stereocenters 2 / 2
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of LASCUFLOXACIN MESYLATE

SMILES

CS(O)(=O)=O.COC1=C2N(CCF)C=C(C(O)=O)C(=O)C2=CC(F)=C1N3C[C@@H](F)[C@@H](CNC4CC4)C3

InChI

InChIKey=LLRDGHMAFPAJJT-DFIJPDEKSA-N
InChI=1S/C21H24F3N3O4.CH4O3S/c1-31-20-17-13(19(28)14(21(29)30)9-26(17)5-4-22)6-15(23)18(20)27-8-11(16(24)10-27)7-25-12-2-3-12;1-5(2,3)4/h6,9,11-12,16,25H,2-5,7-8,10H2,1H3,(H,29,30);1H3,(H,2,3,4)/t11-,16+;/m0./s1

HIDE SMILES / InChI

Molecular Formula CH4O3S
Molecular Weight 96.106
Charge 0
Count
Stereochemistry ACHIRAL
Additional Stereochemistry No
Defined Stereocenters 0 / 0
E/Z Centers 0
Optical Activity NONE

Molecular Formula C21H24F3N3O4
Molecular Weight 439.4282
Charge 0
Count
Stereochemistry ABSOLUTE
Additional Stereochemistry No
Defined Stereocenters 2 / 2
E/Z Centers 0
Optical Activity UNSPECIFIED

LASCUFLOXACIN, a fluoroquinolone derivative, is an antibacterial agent with a broad spectrum of activity against various clinical isolates. It is under development for the treatment of respiratory tract infections and community-acquired pneumonia.

Approval Year

PubMed

PubMed

TitleDatePubMed
Substance Class Chemical
Created
by admin
on Sat Dec 16 07:42:57 GMT 2023
Edited
by admin
on Sat Dec 16 07:42:57 GMT 2023
Record UNII
D25Q04AD78
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
LASCUFLOXACIN MESYLATE
Common Name English
3-QUINOLINECARBOXYLIC ACID, 7-((3S,4S)-3-((CYCLOPROPYLAMINO)METHYL)-4-FLUORO-1-PYRROLIDINYL)-6-FLUORO-1-(2-FLUOROETHYL)-1,4-DIHYDRO-8-METHOXY-4-OXO-, METHANESULFONATE (1:1)
Systematic Name English
LASCUFLOXACIN MESILATE
WHO-DD  
Common Name English
Lascufloxacin mesilate [WHO-DD]
Common Name English
Code System Code Type Description
CAS
1433857-41-0
Created by admin on Sat Dec 16 07:42:57 GMT 2023 , Edited by admin on Sat Dec 16 07:42:57 GMT 2023
PRIMARY
FDA UNII
D25Q04AD78
Created by admin on Sat Dec 16 07:42:57 GMT 2023 , Edited by admin on Sat Dec 16 07:42:57 GMT 2023
PRIMARY
PUBCHEM
71569948
Created by admin on Sat Dec 16 07:42:57 GMT 2023 , Edited by admin on Sat Dec 16 07:42:57 GMT 2023
PRIMARY
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