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Details

Stereochemistry ACHIRAL
Molecular Formula C17H20N2O2S
Molecular Weight 316.418
Optical Activity NONE
Defined Stereocenters 0 / 0
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of TINORIDINE

SMILES

CCOC(=O)C1=C(N)SC2=C1CCN(CC3=CC=CC=C3)C2

InChI

InChIKey=PFENFDGYVLAFBR-UHFFFAOYSA-N
InChI=1S/C17H20N2O2S/c1-2-21-17(20)15-13-8-9-19(11-14(13)22-16(15)18)10-12-6-4-3-5-7-12/h3-7H,2,8-11,18H2,1H3

HIDE SMILES / InChI

Molecular Formula C17H20N2O2S
Molecular Weight 316.418
Charge 0
Count
MOL RATIO 1 MOL RATIO (average)
Stereochemistry ACHIRAL
Additional Stereochemistry No
Defined Stereocenters 0 / 0
E/Z Centers 0
Optical Activity NONE

Description

Tinoridine is a non-steroidal anti-inflammatory and analgesic agent. This agent has been proved pharmacologically to show antiedematous and analgesic actions. The mechanism of the anti-inflammatory action of Tinoridine is attributed to its biomembrane stabilizing action particularly on the lysosomes which are related to cell or tissue damage at the time of inflammation through the release of hydrolytic enzymes. Tinoridine may produce gastrointestinal disorders (nausea, loss of appetite, diarrhea, and constipation), vertigo drowsiness, dry mouth and itching.

Originator

Approval Year

Targets

Primary TargetPharmacologyConditionPotency

Conditions

ConditionModalityTargetsHighest PhaseProduct
Palliative
Nonflamin
Primary
Nonflamin
Primary
Nonflamin
Primary
Nonflamin
Primary
Nonflamin

PubMed

Patents

Sample Use Guides

In Vivo Use Guide
1-2 capsules 3 times a day
Route of Administration: Oral
In Vitro Use Guide
30 uM of Tinoridine HCl hydrochloride inhibited the Phospholipase C-induced lysosomal enzyme release from rat liver lysosomes.
Substance Class Chemical
Record UNII
C9Z9ICZ7YR
Record Status Validated (UNII)
Record Version