Dulozafone is an anticonvulsant and anxiolytic agent. Dulozafone was derived from glycine. Neuro-pharmacological experiments had demonstrated that dulozafone shows the same pharmacological activity as benzodiazepines and a good in vivo affinity for the benzodiazepine receptor. Dulozafone is a pro-drug, metabolized in vivo to an active form. One of its putative metabolites could be ortho-chloro-diazepam, which is pharmacologically active. Dulozafone had the same anticonvulsant effect on kindled seizures as diazepam. It is potent inhibitor of convulsions and epileptic discharges of fully kindled rats. Dulozafone exerts their anticonvulsant properties in inhibiting the propagation of the epileptic discharge from amygdala to other cerebral structures, particularly those implicated in the motor generalization, such as the substantia nigra.