U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class
Concept
Record UNII
BCB1002X86
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
TAS-1553
Code English
TAS1553
Preferred Name English
BENZAMIDE, 5-CHLORO-2-((((1S,2R)-1-(4,5-DIHYDRO-5-OXO-1,3,4-OXADIAZOL-2-YL)-2-(6-FLUORO-2,3-DIMETHYLPHENYL)PROPYL)AMINO)SULFONYL)-
Systematic Name English
Code System Code Type Description
NCI_THESAURUS
C176434
Created by admin on Wed Apr 02 06:43:58 GMT 2025 , Edited by admin on Wed Apr 02 06:43:58 GMT 2025
PRIMARY
FDA UNII
BCB1002X86
Created by admin on Wed Apr 02 06:43:58 GMT 2025 , Edited by admin on Wed Apr 02 06:43:58 GMT 2025
PRIMARY
PUBCHEM
132203319
Created by admin on Wed Apr 02 06:43:58 GMT 2025 , Edited by admin on Wed Apr 02 06:43:58 GMT 2025
PRIMARY
CAS
2166023-31-8
Created by admin on Wed Apr 02 06:43:58 GMT 2025 , Edited by admin on Wed Apr 02 06:43:58 GMT 2025
PRIMARY
This is a non-substance concept
Related Record Type Details
SALT/SOLVATE -> PARENT
TARGET -> INHIBITOR
RNR activity was determined by its ability to reduce cytidine diphosphate (CDP) to deoxycytidine diphosphate (dCDP), based on a previous report
IC50
TARGET -> INHIBITOR
Targets protein-protein interaction between R1 and R2.
Kd
Related Record Type Details
ACTIVE MOIETY
This is a non-substance concept