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Details

Stereochemistry ACHIRAL
Molecular Formula C10H14ClN3OS
Molecular Weight 259.756
Optical Activity NONE
Defined Stereocenters 0 / 0
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of AZINTAMIDE

SMILES

CCN(CC)C(=O)CSC1=NN=C(Cl)C=C1

InChI

InChIKey=SSLKKMZJCJBOML-UHFFFAOYSA-N
InChI=1S/C10H14ClN3OS/c1-3-14(4-2)10(15)7-16-9-6-5-8(11)12-13-9/h5-6H,3-4,7H2,1-2H3

HIDE SMILES / InChI

Molecular Formula C10H14ClN3OS
Molecular Weight 259.756
Charge 0
Count
Stereochemistry ACHIRAL
Additional Stereochemistry No
Defined Stereocenters 0 / 0
E/Z Centers 0
Optical Activity NONE

Azintamide was initially studied as a therapeutic agent in psoriasis vulgaris. Then was shown, the drug was effective and safe in the treatment of patients with dyspepsia symptoms by the modulation of visceral sensitivity and/or gastrointestinal motility.

Approval Year

Conditions

Conditions

ConditionModalityTargetsHighest PhaseProduct
Primary
Unknown

Approved Use

Unknown
PubMed

PubMed

TitleDatePubMed
[Azintamid as a therapeutic agent in psoriasis vulgaris - a therapeutic study].
1983
Gas-liquid chromatographic determination of azintamide (Ora-gallin) in pharmaceutical formulations.
1985 May 24
[Efficacy and safety of compound azintamide on dyspepsia symptoms in a multicentre self-controlled trial].
2008 Nov

Sample Use Guides

Two tablets of compound azintamide were administered orally following a meal, tid for 2 weeks
Route of Administration: Oral
Substance Class Chemical
Created
by admin
on Sat Dec 16 16:31:40 GMT 2023
Edited
by admin
on Sat Dec 16 16:31:40 GMT 2023
Record UNII
ACZ6L64B41
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
AZINTAMIDE
INN   MART.   MI   WHO-DD  
INN  
Official Name English
2-((6-CHLORO-3-PYRIDAZINYL)THIO)-N,N-DIETHYLACETAMIDE
Systematic Name English
NSC-291837
Code English
Azintamide [WHO-DD]
Common Name English
ST 9067
Code English
AZINTAMIDE [MART.]
Common Name English
AZINTAMIDE [MI]
Common Name English
AZINTHIAMIDE
Common Name English
COLERIN
Brand Name English
azintamide [INN]
Common Name English
ST-9067
Code English
Classification Tree Code System Code
NCI_THESAURUS C66913
Created by admin on Sat Dec 16 16:31:40 GMT 2023 , Edited by admin on Sat Dec 16 16:31:40 GMT 2023
Code System Code Type Description
PUBCHEM
71105
Created by admin on Sat Dec 16 16:31:40 GMT 2023 , Edited by admin on Sat Dec 16 16:31:40 GMT 2023
PRIMARY
FDA UNII
ACZ6L64B41
Created by admin on Sat Dec 16 16:31:40 GMT 2023 , Edited by admin on Sat Dec 16 16:31:40 GMT 2023
PRIMARY
DRUG BANK
DB13992
Created by admin on Sat Dec 16 16:31:40 GMT 2023 , Edited by admin on Sat Dec 16 16:31:40 GMT 2023
PRIMARY
NSC
291837
Created by admin on Sat Dec 16 16:31:40 GMT 2023 , Edited by admin on Sat Dec 16 16:31:40 GMT 2023
PRIMARY
SMS_ID
100000086085
Created by admin on Sat Dec 16 16:31:40 GMT 2023 , Edited by admin on Sat Dec 16 16:31:40 GMT 2023
PRIMARY
ECHA (EC/EINECS)
217-384-2
Created by admin on Sat Dec 16 16:31:40 GMT 2023 , Edited by admin on Sat Dec 16 16:31:40 GMT 2023
PRIMARY
EPA CompTox
DTXSID50171370
Created by admin on Sat Dec 16 16:31:40 GMT 2023 , Edited by admin on Sat Dec 16 16:31:40 GMT 2023
PRIMARY
DRUG CENTRAL
275
Created by admin on Sat Dec 16 16:31:40 GMT 2023 , Edited by admin on Sat Dec 16 16:31:40 GMT 2023
PRIMARY
EVMPD
SUB05658MIG
Created by admin on Sat Dec 16 16:31:40 GMT 2023 , Edited by admin on Sat Dec 16 16:31:40 GMT 2023
PRIMARY
INN
2063
Created by admin on Sat Dec 16 16:31:40 GMT 2023 , Edited by admin on Sat Dec 16 16:31:40 GMT 2023
PRIMARY
MERCK INDEX
m1019
Created by admin on Sat Dec 16 16:31:40 GMT 2023 , Edited by admin on Sat Dec 16 16:31:40 GMT 2023
PRIMARY Merck Index
NCI_THESAURUS
C74232
Created by admin on Sat Dec 16 16:31:40 GMT 2023 , Edited by admin on Sat Dec 16 16:31:40 GMT 2023
PRIMARY
CAS
1830-32-6
Created by admin on Sat Dec 16 16:31:40 GMT 2023 , Edited by admin on Sat Dec 16 16:31:40 GMT 2023
PRIMARY
ChEMBL
CHEMBL2104678
Created by admin on Sat Dec 16 16:31:40 GMT 2023 , Edited by admin on Sat Dec 16 16:31:40 GMT 2023
PRIMARY
RXCUI
402580
Created by admin on Sat Dec 16 16:31:40 GMT 2023 , Edited by admin on Sat Dec 16 16:31:40 GMT 2023
PRIMARY RxNorm
Related Record Type Details
ACTIVE MOIETY