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Details

Stereochemistry ACHIRAL
Molecular Formula C19H20N2
Molecular Weight 276.3755
Optical Activity NONE
Defined Stereocenters 0 / 0
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of MEBHYDROLIN

SMILES

CN1CCC2=C(C1)C3=C(C=CC=C3)N2CC4=CC=CC=C4

InChI

InChIKey=FQQIIPAOSKSOJM-UHFFFAOYSA-N
InChI=1S/C19H20N2/c1-20-12-11-19-17(14-20)16-9-5-6-10-18(16)21(19)13-15-7-3-2-4-8-15/h2-10H,11-14H2,1H3

HIDE SMILES / InChI

Molecular Formula C19H20N2
Molecular Weight 276.3755
Charge 0
Count
MOL RATIO 1 MOL RATIO (average)
Stereochemistry ACHIRAL
Additional Stereochemistry No
Defined Stereocenters 0 / 0
E/Z Centers 0
Optical Activity NONE

Description

Mebhydrolin (INN) or mebhydroline is a histamine H1-receptor antagonist. It is not available in the United States, but it is available in various other countries under the brand names Bexidal and Diazolin. It is used for symptomatic relief of allergic symptoms caused by histamine release, including nasal allergies and allergic dermatosis.

Approval Year

Targets

Primary TargetPharmacologyConditionPotency

Conditions

ConditionModalityTargetsHighest PhaseProduct
Primary
Bexidal
Primary
Bexidal
Primary
Bexidal
Primary
Bexidal

Doses

AEs

PubMed

Sample Use Guides

In Vivo Use Guide
Adults and children over 10 years 2-6 tablets daily Children from 5-10 years 2-4 tablets daily Children from 2-5 years 1-3 tablets daily Children up to 2 years 1-2 tablets daily Treatment should be given in several single doses daily.
Route of Administration: Oral
In Vitro Use Guide
Unknown
Substance Class Chemical
Record UNII
9SUK9B7XVY
Record Status Validated (UNII)
Record Version