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Details

Stereochemistry ACHIRAL
Molecular Formula C15H16N4O
Molecular Weight 268.3137
Optical Activity NONE
Defined Stereocenters 0 / 0
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of RIPAZEPAM

SMILES

CCN1N=C(C)C2=C1C(=NCC(=O)N2)C3=CC=CC=C3

InChI

InChIKey=YFHYNLHGFKXAIQ-UHFFFAOYSA-N
InChI=1S/C15H16N4O/c1-3-19-15-13(10(2)18-19)17-12(20)9-16-14(15)11-7-5-4-6-8-11/h4-8H,3,9H2,1-2H3,(H,17,20)

HIDE SMILES / InChI

Molecular Formula C15H16N4O
Molecular Weight 268.3137
Charge 0
Count
MOL RATIO 1 MOL RATIO (average)
Stereochemistry ACHIRAL
Additional Stereochemistry No
Defined Stereocenters 0 / 0
E/Z Centers 0
Optical Activity NONE

Description

Ripazepam (CI 683 or pyrazapon) is a pyrazolodiazepine that has anxiolytic effects. It is related to certain benzodiazepines such as zolazepam. In animal studies, it showed anxiolytic effects without sedative or depressant effects. In rats, it did not elicit a tumorigenic potential. Although ripazepam was found significantly superior to placebo and was well tolerated in neurotic patients, it has never been marketed for clinical use.

Approval Year

Substance Class Chemical
Record UNII
92000WH9C9
Record Status Validated (UNII)
Record Version