RIPAZEPAM

Details

Stereochemistry	ACHIRAL
Molecular Formula	C15H16N4O
Molecular Weight	268.3137
Optical Activity	NONE
Defined Stereocenters	0 / 0
E/Z Centers	0
Charge	0

SHOW SMILES / InChI

Structure Search

SMILES

CCN1N=C(C)C2=C1C(=NCC(=O)N2)C3=CC=CC=C3

InChI

InChIKey=YFHYNLHGFKXAIQ-UHFFFAOYSA-N

InChI=1S/C15H16N4O/c1-3-19-15-13(10(2)18-19)17-12(20)9-16-14(15)11-7-5-4-6-8-11/h4-8H,3,9H2,1-2H3,(H,17,20)

HIDE SMILES / InChI

Molecular Formula	C15H16N4O
Molecular Weight	268.3137
Charge	0
Count

Stereochemistry	ACHIRAL
Additional Stereochemistry	No
Defined Stereocenters	0 / 0
E/Z Centers	0
Optical Activity	NONE

Description
Sources: http://www.inchem.org/documents/iarc/vol66/ripazepam.html | https://www.ncbi.nlm.nih.gov/pubmed/6724192 | https://www.ncbi.nlm.nih.gov/pubmed/780378

Ripazepam (CI 683 or pyrazapon) is a pyrazolodiazepine that has anxiolytic effects. It is related to certain benzodiazepines such as zolazepam. In animal studies, it showed anxiolytic effects without sedative or depressant effects. In rats, it did not elicit a tumorigenic potential. Although ripazepam was found significantly superior to placebo and was well tolerated in neurotic patients, it has never been marketed for clinical use.

Approval Year

Patents

Substance Class	Chemical Created by `admin` on `Fri Dec 15 15:20:20 UTC 2023` Edited by `admin` on `Fri Dec 15 15:20:20 UTC 2023`
Record UNII	92000WH9C9
Record Status	`Validated (UNII)`
Record Version

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Name

Type

Language

RIPAZEPAM

Official Name

English

1-Ethyl-4,6-dihydro-3-methyl-8-phenylpyrazolo[4,3-E][1,4]diazepin-5(1H)-one

Systematic Name

English

CL-683

Code

English

RIPAZEPAM [USAN]

Common Name

English

PYRAZOLO(4,3-E)(1,4)DIAZEPIN-5(1H)-ONE, 1-ETHYL-4,6-DIHYDRO-3-METHYL-8-PHENYL-

Systematic Name

English

RIPAZEPAM [IARC]

Common Name

English

ripazepam [INN]

Common Name

English

Classification Tree Code System Code

NCI_THESAURUS

C1012