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Details

Stereochemistry RACEMIC
Molecular Formula C10H15N
Molecular Weight 149.2328
Optical Activity ( + / - )
Defined Stereocenters 0 / 1
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of PHENPROMETHAMINE

SMILES

CNCC(C)C1=CC=CC=C1

InChI

InChIKey=AUFSOOYCQYDGES-UHFFFAOYSA-N
InChI=1S/C10H15N/c1-9(8-11-2)10-6-4-3-5-7-10/h3-7,9,11H,8H2,1-2H3

HIDE SMILES / InChI
Molecular Formula C10H15N
Molecular Weight 149.2328
Charge 0
Count
MOL RATIO 1 MOL RATIO (average)
Stereochemistry RACEMIC
Additional Stereochemistry No
Defined Stereocenters 0 / 1
E/Z Centers 0
Optical Activity ( + / - )

Description

Phenpromethamine is an adrenergic agent. Phenpromethamine was used as vasodilator agent. It is a stimulant which is banned in sport. It is available in supplements which are sold as fat burners or pre-workout boosters. Phenpromethamine is a potent CYP2D6 inhibitor.

Approval Year

1943
64

Overview

CYP3A4CYP2C9CYP2D6hERG
inhibitor
1,587
inhibitor
1,852

OverviewOther

Other InhibitorOther SubstrateOther Inducer

Drug as perpetrator​

PubMed

Substance Class Chemical
Record UNII
7D4542I59V
Record Status Validated (UNII)
Record Version
NIH
NCATS
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