ALLYLPRODINE

U.S. Department of Health & Human Services Divider Arrow

National Institutes of Health Divider Arrow

NCATS

Description
Sources: https://www.ncbi.nlm.nih.gov/pubmed/13412197 | https://www.ncbi.nlm.nih.gov/pubmed/1246054 | https://www.deadiversion.usdoj.gov/fed_regs/quotas/2014/fr0825.htm

Allylprodine (Ro 2-7113) is an opioid analgesic. It is stereoselective, with one isomer being much more active. Allylprodine is included in Schedule I of the US Controlled Substances Act 1970 as a Narcotic with ACSCN 9602 and a 2014 annual aggregate manufacturing quota of 2 grammes.

Originator

Approval Year

PubMed

PubMed

Title	Date	PubMed
Allylprodine analogues as receptor probes. Evidence that phenolic and nonphenolic ligands interact with different subsites on identical opioid receptors.	1981-07	6268787
Conformation of 2,9-dimethyl-3'-hydroxy-5-phenyl-6,7-genzomorphan and its relation to other analgetics and enkephalin.	1978-07	209186
Stereochemical studies on medicinal agents. 19. X-ray crystal structures of two (+/-)-allylprodine diastereomers. The role of the allyl group in conferring high stereoselectivity and potency at analgetic receptors.	1976-01	1246054
Analgesic activity and toxicity of Ro 2-7113.	1957-01-01	13412197

Patents

Patents

Substance Class	Mixture Created by `admin` on `Mon Mar 31 18:18:47 GMT 2025` Edited by `admin` on `Mon Mar 31 18:18:47 GMT 2025`
Record UNII	4343OEZ18O
Record Status	`Validated (UNII)`
Record Version

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Name

Type

Language

ACSCN-9602

Preferred Name

English

ALLYLPRODINE

Official Name

English

3-ALLYL-1-METHYL-4-PHENYL-4-PROPIONYLOXYPIPERIDINE

Common Name

English

ALPERIDINE

Common Name

English

allylprodine [INN]

Common Name

English

DEA NO. 9602

Code

English

NIH-7440

Code

English

IDS-NA-007

Code

English

ALLYLPRODINE [MI]

Common Name

English

RO 2-7113

Common Name

English

Classification Tree Code System Code

NCI_THESAURUS

C241

Created by admin on Mon Mar 31 18:18:47 GMT 2025 , Edited by admin on Mon Mar 31 18:18:47 GMT 2025

DEA NO.

9602

Created by admin on Mon Mar 31 18:18:47 GMT 2025 , Edited by admin on Mon Mar 31 18:18:47 GMT 2025

Code System Code Type Description

INN

891

Created by admin on Mon Mar 31 18:18:47 GMT 2025 , Edited by admin on Mon Mar 31 18:18:47 GMT 2025

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EPA CompTox

DTXSID80865210

Created by admin on Mon Mar 31 18:18:47 GMT 2025 , Edited by admin on Mon Mar 31 18:18:47 GMT 2025

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ChEMBL

CHEMBL2103995

Created by admin on Mon Mar 31 18:18:47 GMT 2025 , Edited by admin on Mon Mar 31 18:18:47 GMT 2025

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MERCK INDEX

m1557

Created by admin on Mon Mar 31 18:18:47 GMT 2025 , Edited by admin on Mon Mar 31 18:18:47 GMT 2025

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Merck Index

NCI_THESAURUS

C72102

Created by admin on Mon Mar 31 18:18:47 GMT 2025 , Edited by admin on Mon Mar 31 18:18:47 GMT 2025

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DRUG BANK

DB01542

Created by admin on Mon Mar 31 18:18:47 GMT 2025 , Edited by admin on Mon Mar 31 18:18:47 GMT 2025

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PUBCHEM

32938

Created by admin on Mon Mar 31 18:18:47 GMT 2025 , Edited by admin on Mon Mar 31 18:18:47 GMT 2025

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FDA UNII

4343OEZ18O

Created by admin on Mon Mar 31 18:18:47 GMT 2025 , Edited by admin on Mon Mar 31 18:18:47 GMT 2025

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WIKIPEDIA

ALLYLPRODINE

Created by admin on Mon Mar 31 18:18:47 GMT 2025 , Edited by admin on Mon Mar 31 18:18:47 GMT 2025

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CAS

25384-17-2

Created by admin on Mon Mar 31 18:18:47 GMT 2025 , Edited by admin on Mon Mar 31 18:18:47 GMT 2025

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EVMPD

SUB05340MIG

Created by admin on Mon Mar 31 18:18:47 GMT 2025 , Edited by admin on Mon Mar 31 18:18:47 GMT 2025

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SMS_ID

100000087438

Created by admin on Mon Mar 31 18:18:47 GMT 2025 , Edited by admin on Mon Mar 31 18:18:47 GMT 2025

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All of the following components must be present:


					G98M360H09

ALLYLPRODINE, .ALPHA.-


					028U1A6J7B

ALLYLPRODINE, .BETA.-

Related Record Type Details


					WF82M29MCG

ALLYLPRODINE HYDROCHLORIDE, .BETA.-

SALT/SOLVATE -> PARENT

Comments:

APPROXIMATE PURE ANHYDROUS DRUG CONTENT (IN PERCENT)

Amount:

Related Record Type Details


					4343OEZ18O

ACTIVE MOIETY

Definition References