ALLYLPRODINE

Description
Sources: https://www.ncbi.nlm.nih.gov/pubmed/13412197 | https://www.ncbi.nlm.nih.gov/pubmed/1246054 | https://www.deadiversion.usdoj.gov/fed_regs/quotas/2014/fr0825.htm

Allylprodine (Ro 2-7113) is an opioid analgesic. It is stereoselective, with one isomer being much more active. Allylprodine is included in Schedule I of the US Controlled Substances Act 1970 as a Narcotic with ACSCN 9602 and a 2014 annual aggregate manufacturing quota of 2 grammes.

Originator

Approval Year

PubMed

Title	Date	PubMed
Analgesic activity and toxicity of Ro 2-7113.	1957 Jan 1	13412197
Stereochemical studies on medicinal agents. 19. X-ray crystal structures of two (+/-)-allylprodine diastereomers. The role of the allyl group in conferring high stereoselectivity and potency at analgetic receptors.	1976 Jan	1246054
Conformation of 2,9-dimethyl-3'-hydroxy-5-phenyl-6,7-genzomorphan and its relation to other analgetics and enkephalin.	1978 Jul	209186
Allylprodine analogues as receptor probes. Evidence that phenolic and nonphenolic ligands interact with different subsites on identical opioid receptors.	1981 Jul	6268787

Patents

Substance Class	Mixture Created by `admin` on `Fri Dec 15 16:05:44 GMT 2023` Edited by `admin` on `Fri Dec 15 16:05:44 GMT 2023`
Record UNII	4343OEZ18O
Record Status	`Validated (UNII)`
Record Version

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Name

Type

Language

ALLYLPRODINE

Official Name

English

3-ALLYL-1-METHYL-4-PHENYL-4-PROPIONYLOXYPIPERIDINE

Common Name

English

ACSCN-9602

Code

English

ALPERIDINE

Common Name

English

allylprodine [INN]

Common Name

English

DEA NO. 9602

Code

English

NIH-7440

Code

English

IDS-NA-007

Code

English

ALLYLPRODINE [MI]

Common Name

English

RO 2-7113

Common Name

English

Classification Tree Code System Code

NCI_THESAURUS

C241