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Details

Stereochemistry RACEMIC
Molecular Formula C9H14N2
Molecular Weight 150.2209
Optical Activity ( + / - )
Defined Stereocenters 0 / 1
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of PHENIPRAZINE

SMILES

CC(CC1=CC=CC=C1)NN

InChI

InChIKey=VXTWEDPZMSVFEF-UHFFFAOYSA-N
InChI=1S/C9H14N2/c1-8(11-10)7-9-5-3-2-4-6-9/h2-6,8,11H,7,10H2,1H3

HIDE SMILES / InChI

Molecular Formula C9H14N2
Molecular Weight 150.2209
Charge 0
Count
MOL RATIO 1 MOL RATIO (average)
Stereochemistry RACEMIC
Additional Stereochemistry No
Defined Stereocenters 0 / 1
E/Z Centers 0
Optical Activity ( + / - )

Description

PHENIPRAZINE is a monoamine oxidase inhibitor of the hydrazine chemical class that was used for the treatment of depression, schizophrenia, and also as a long-acting coronary vasodilator in patients suffering from angina pectoris. PHENIPRAZINE was discontinued due to toxicity concerns such as jaundice, amblyopia, and optic neuritis.

Approval Year

Targets

Primary TargetPharmacologyConditionPotency

Conditions

ConditionModalityTargetsHighest PhaseProduct
Primary
Catron
Primary
Catron

Doses

AEs

Sourcing

PubMed

Substance Class Chemical
Record UNII
37VKD7067M
Record Status Validated (UNII)
Record Version