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Details

Stereochemistry RACEMIC
Molecular Formula C12H17NO3
Molecular Weight 223.2683
Optical Activity ( + / - )
Defined Stereocenters 2 / 2
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of RIMITEROL

SMILES

[H][C@]1(CCCCN1)[C@H](O)C2=CC(O)=C(O)C=C2

InChI

InChIKey=IYMMESGOJVNCKV-JOYOIKCWSA-N
InChI=1S/C12H17NO3/c14-10-5-4-8(7-11(10)15)12(16)9-3-1-2-6-13-9/h4-5,7,9,12-16H,1-3,6H2/t9-,12+/m0/s1

HIDE SMILES / InChI

Molecular Formula C12H17NO3
Molecular Weight 223.2683
Charge 0
Count
Stereochemistry ABSOLUTE
Additional Stereochemistry No
Defined Stereocenters 2 / 2
E/Z Centers 0
Optical Activity UNSPECIFIED

Rimiterol is erythro-(3,4-dihydroxyphenyl)-2-piperidyl-methanol hydrobromide, and is a catecholamine. It is a selective β2-adrenoreceptor agonist, but is not effective as a bronchodilator by the oral route of administration. Rimiterol is available at present as an aerosol, though preliminary studies suggest that it may be of value in the intravenous therapy of severe asthma.

Approval Year

Patents

Patents

Sample Use Guides

As metered-dose aerosol: 250-500 mcg when needed. Max: 8 times/24 hr. Not to repeat dose in <1 hr.
Route of Administration: Respiratory
Substance Class Chemical
Created
by admin
on Fri Dec 15 15:26:40 GMT 2023
Edited
by admin
on Fri Dec 15 15:26:40 GMT 2023
Record UNII
26GIW6ZLPH
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
RIMITEROL
INN   MI   WHO-DD  
INN  
Official Name English
RIMITEROL [MI]
Common Name English
Rimiterol [WHO-DD]
Common Name English
rimiterol [INN]
Common Name English
2-PIPERIDINEMETHANOL, .ALPHA.-(3,4-DIHYDROXYPHENYL)-, (R*,S*)-
Systematic Name English
Classification Tree Code System Code
WHO-VATC QR03AC05
Created by admin on Fri Dec 15 15:26:40 GMT 2023 , Edited by admin on Fri Dec 15 15:26:40 GMT 2023
WHO-ATC R03AC05
Created by admin on Fri Dec 15 15:26:40 GMT 2023 , Edited by admin on Fri Dec 15 15:26:40 GMT 2023
NCI_THESAURUS C48149
Created by admin on Fri Dec 15 15:26:40 GMT 2023 , Edited by admin on Fri Dec 15 15:26:40 GMT 2023
Code System Code Type Description
EVMPD
SUB10324MIG
Created by admin on Fri Dec 15 15:26:40 GMT 2023 , Edited by admin on Fri Dec 15 15:26:40 GMT 2023
PRIMARY
CAS
32953-89-2
Created by admin on Fri Dec 15 15:26:40 GMT 2023 , Edited by admin on Fri Dec 15 15:26:40 GMT 2023
PRIMARY
ChEMBL
CHEMBL1097630
Created by admin on Fri Dec 15 15:26:40 GMT 2023 , Edited by admin on Fri Dec 15 15:26:40 GMT 2023
PRIMARY
RXCUI
9388
Created by admin on Fri Dec 15 15:26:40 GMT 2023 , Edited by admin on Fri Dec 15 15:26:40 GMT 2023
PRIMARY RxNorm
EPA CompTox
DTXSID70186603
Created by admin on Fri Dec 15 15:26:40 GMT 2023 , Edited by admin on Fri Dec 15 15:26:40 GMT 2023
PRIMARY
NCI_THESAURUS
C81639
Created by admin on Fri Dec 15 15:26:40 GMT 2023 , Edited by admin on Fri Dec 15 15:26:40 GMT 2023
PRIMARY
FDA UNII
26GIW6ZLPH
Created by admin on Fri Dec 15 15:26:40 GMT 2023 , Edited by admin on Fri Dec 15 15:26:40 GMT 2023
PRIMARY
PUBCHEM
46886609
Created by admin on Fri Dec 15 15:26:40 GMT 2023 , Edited by admin on Fri Dec 15 15:26:40 GMT 2023
PRIMARY
DRUG CENTRAL
2385
Created by admin on Fri Dec 15 15:26:40 GMT 2023 , Edited by admin on Fri Dec 15 15:26:40 GMT 2023
PRIMARY
WIKIPEDIA
RIMITEROL
Created by admin on Fri Dec 15 15:26:40 GMT 2023 , Edited by admin on Fri Dec 15 15:26:40 GMT 2023
PRIMARY
MESH
C084590
Created by admin on Fri Dec 15 15:26:40 GMT 2023 , Edited by admin on Fri Dec 15 15:26:40 GMT 2023
PRIMARY
SMS_ID
100000080567
Created by admin on Fri Dec 15 15:26:40 GMT 2023 , Edited by admin on Fri Dec 15 15:26:40 GMT 2023
PRIMARY
INN
3121
Created by admin on Fri Dec 15 15:26:40 GMT 2023 , Edited by admin on Fri Dec 15 15:26:40 GMT 2023
PRIMARY
DRUG BANK
DB13559
Created by admin on Fri Dec 15 15:26:40 GMT 2023 , Edited by admin on Fri Dec 15 15:26:40 GMT 2023
PRIMARY
ECHA (EC/EINECS)
251-305-2
Created by admin on Fri Dec 15 15:26:40 GMT 2023 , Edited by admin on Fri Dec 15 15:26:40 GMT 2023
PRIMARY
MERCK INDEX
m9623
Created by admin on Fri Dec 15 15:26:40 GMT 2023 , Edited by admin on Fri Dec 15 15:26:40 GMT 2023
PRIMARY Merck Index
Related Record Type Details
SALT/SOLVATE -> PARENT
Related Record Type Details
ACTIVE MOIETY