Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Sat Dec 16 12:11:01 GMT 2023
by
admin
on
Sat Dec 16 12:11:01 GMT 2023
|
| Protein Sub Type | |
| Sequence Type | COMPLETE |
| Record UNII |
1AG1A6ENX6
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
1AG1A6ENX6
Created by
admin on Sat Dec 16 12:11:02 GMT 2023 , Edited by admin on Sat Dec 16 12:11:02 GMT 2023
|
PRIMARY |
| From | To |
|---|---|
| 1_155 | 1_231 |
| Glycosylation Type | HUMAN |
| Glycosylation Link Type | Site |
|---|---|
| N | 1_5 |
| N | 1_66 |
| Related Record | Type | Details | ||
|---|---|---|---|---|
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AGONIST -> TARGET | |||
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INHIBITOR -> TARGET | |||
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AGONIST -> TARGET |
Ki
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INHIBITOR -> TARGET |
Ki
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
INHIBITOR
Ki
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AGONIST -> TARGET |
In vitro binding assays revealed that RA-7 possessed higher 5-HT7 receptor affinity than LP-211 and a better selectivity profile over a panel of 5-HT receptor subtypes.
ANTAGONIST
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TARGET -> AGONIST |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
INHIBITOR
Ki
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INHIBITOR -> TARGET |
Ki
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INHIBITOR -> TARGET | |||
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AGONIST -> TARGET |
Eletriptan binds with high affinity to 5-HT1B, 5-HT1D and 5-HT1F receptors, has modest affinity for 5-HT1A, 5-HT1E, 5-HT2B and 5-HT7 receptors
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INHIBITOR -> TARGET |
ANTAGONIST
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AGONIST -> TARGET | |||
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AGONIST -> TARGET | |||
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INHIBITOR -> TARGET |
Cell:SF9; ligand:3H-5-ct
BINDING
Ki
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AGONIST -> TARGET |
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AGONIST -> TARGET |
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INHIBITOR -> TARGET | |||
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AGONIST -> TARGET |
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| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT | CHEMICAL |
|