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Details

Stereochemistry ACHIRAL
Molecular Formula C19H20ClN3O
Molecular Weight 341.835
Optical Activity NONE
Defined Stereocenters 0 / 0
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of SARIPIDEM

SMILES

CCCC(=O)N(C)CC1=C(N=C2C=CC=CN12)C3=CC=C(Cl)C=C3

InChI

InChIKey=LIFDPEORUVTOCP-UHFFFAOYSA-N
InChI=1S/C19H20ClN3O/c1-3-6-18(24)22(2)13-16-19(14-8-10-15(20)11-9-14)21-17-7-4-5-12-23(16)17/h4-5,7-12H,3,6,13H2,1-2H3

HIDE SMILES / InChI

Molecular Formula C19H20ClN3O
Molecular Weight 341.835
Charge 0
Count
MOL RATIO 1 MOL RATIO (average)
Stereochemistry ACHIRAL
Additional Stereochemistry No
Defined Stereocenters 0 / 0
E/Z Centers 0
Optical Activity NONE

Description

Synthélabo developed a saripidem (also known as SL 850274) as a potential anxiolytic agent that modulates the benzodiazepine-binding site on GABAA receptor via primary binding with ω1 subtype. Saripidem was studied in phase II clinical trials for the treatment of patients with anxiety disorders. However, information about the further development of the drug is not available.

Originator

Approval Year

PubMed

Substance Class Chemical
Record UNII
0J6174G60N
Record Status Validated (UNII)
Record Version