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Details

Stereochemistry RACEMIC
Molecular Formula C11H25N.ClH
Molecular Weight 207.784
Optical Activity ( + / - )
Defined Stereocenters 0 / 1
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of IPROHEPTINE HYDROCHLORIDE

SMILES

Cl.CC(C)CCCC(C)NC(C)C

InChI

InChIKey=QYEORIIWGAAORG-UHFFFAOYSA-N
InChI=1S/C11H25N.ClH/c1-9(2)7-6-8-11(5)12-10(3)4;/h9-12H,6-8H2,1-5H3;1H

HIDE SMILES / InChI

Description

Iproheptine (Metron, Susat) is a vasoconstrictor, antihistamine, nasal decongestant marketed in Japan.

CNS Activity

CNS Active
3,913

Approval Year

Unknown
139,594

Targets

Primary TargetPharmacologyConditionPotency
Histamine H1 receptor
315
Antagonist
2,778

Conditions

ConditionModalityTargetsHighest PhaseProduct
Nasal congestion
26
 Primary
Approved
8,429
METRON

Sample Use Guides

In Vivo Use Guide
Maximum daily dose - 150mg
Route of Administration: Oral
In Vitro Use Guide
Unknown
ACTIVE MOIETY
Structure of IPROHEPTINE
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