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Details

Stereochemistry ACHIRAL
Molecular Formula C15H17N5S
Molecular Weight 299.394
Optical Activity NONE
Defined Stereocenters 0 / 0
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of PENTIAPINE

SMILES

CN1CCN(CC1)C2=NC3=CC=CC=C3SC4=NC=CN24

InChI

InChIKey=FACMWMBWGSPRKO-UHFFFAOYSA-N
InChI=1S/C15H17N5S/c1-18-8-10-19(11-9-18)14-17-12-4-2-3-5-13(12)21-15-16-6-7-20(14)15/h2-7H,8-11H2,1H3

HIDE SMILES / InChI

Description

Pentiapine is a dopamine release inhibitor. It is a tranquiliser. Pentiapine produces a dose-dependent decrease in spontaneous motor activity and blocks the morphineinduced hyperactivity. Moreover, this drug in itself has no effect on place conditioning but blocks the acquisition of morphine-induced conditioned place preference.

Approval Year

PubMed

Sample Use Guides

In Vivo Use Guide
24 and 32 mg/kg
Route of Administration: Intraperitoneal