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Details

Stereochemistry ACHIRAL
Molecular Formula C12H13BrN4O2S
Molecular Weight 357.226
Optical Activity NONE
Defined Stereocenters 0 / 0
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of SULFABROMOMETHAZINE

SMILES

CC1=NC(NS(=O)(=O)C2=CC=C(N)C=C2)=NC(C)=C1Br

InChI

InChIKey=KWXCNODTHBHSIQ-UHFFFAOYSA-N
InChI=1S/C12H13BrN4O2S/c1-7-11(13)8(2)16-12(15-7)17-20(18,19)10-5-3-9(14)4-6-10/h3-6H,14H2,1-2H3,(H,15,16,17)

HIDE SMILES / InChI

Description

Sulfabromomethazine is a long-acting derivative of sulfamezathine that is used in the poultry, swine and cattle industries for the treatment of coccidiosis and various bacterial infections. Single oral doses of the drug have been used to treat calf diphteria and pneumonia, metritis, foot root and septic mastitis in cattle with repeated dose 48 hors later sometimes required. Use of sulfabromomethazine during the last 3 months of pregnancy should be avoided. The compound is now rarely used.

Originator

Approval Year

Targets

Primary TargetPharmacologyConditionPotency
230.0 µM [IC50]

Conditions

ConditionModalityTargetsHighest PhaseProduct
Curative
Sulfabrom
Curative
Sulfabrom

PubMed

Sample Use Guides

In Vivo Use Guide
Unknown
Route of Administration: Oral
In Vitro Use Guide
Unknown