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Details

Stereochemistry RACEMIC
Molecular Formula C12H17NO3.BrH
Molecular Weight 304.18
Optical Activity ( + / - )
Defined Stereocenters 2 / 2
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of RIMITEROL HYDROBROMIDE

SMILES

Br.[H][C@]1(CCCCN1)[C@H](O)C2=CC(O)=C(O)C=C2

InChI

InChIKey=QPYZEEKXUYXZBK-PKKHVXKMSA-N
InChI=1S/C12H17NO3.BrH/c14-10-5-4-8(7-11(10)15)12(16)9-3-1-2-6-13-9;/h4-5,7,9,12-16H,1-3,6H2;1H/t9-,12+;/m0./s1

HIDE SMILES / InChI
Rimiterol is erythro-(3,4-dihydroxyphenyl)-2-piperidyl-methanol hydrobromide, and is a catecholamine. It is a selective β2-adrenoreceptor agonist, but is not effective as a bronchodilator by the oral route of administration. Rimiterol is available at present as an aerosol, though preliminary studies suggest that it may be of value in the intravenous therapy of severe asthma.

Approval Year

Patents

Patents

Sample Use Guides

As metered-dose aerosol: 250-500 mcg when needed. Max: 8 times/24 hr. Not to repeat dose in <1 hr.
Route of Administration: Respiratory
Name Type Language
RIMITEROL HYDROBROMIDE
MART.   MI   USAN   WHO-DD  
USAN  
Official Name English
2-PIPERIDINEMETHANOL, .ALPHA.-(3,4-DIHYDROXYPHENYL)-, (R*,S*)-, HBR
Common Name English
WG-253
Code English
RIMITEROL HYDROBROMIDE [MART.]
Common Name English
R 798
Code English
NSC-289336
Code English
PULMADIL
Brand Name English
Rimiterol hydrobromide [WHO-DD]
Common Name English
RIMITEROL HYDROBROMIDE [MI]
Common Name English
R-798
Code English
2-PIPERIDINEMETHANOL, .ALPHA.-(3,4-DIHYDROXYPHENYL)-, (R*,S*)-, HYDROBROMIDE
Systematic Name English
erythro-α-(3,4-Dihydroxyphenyl)-2-piperidinemethanol hydrobromide
Common Name English
RIMITEROL HYDROBROMIDE [USAN]
Common Name English
ERYTHRO-.ALPHA.-(3,4-DIHYDROXYPHENYL)-2-PIPERIDINEMETHANOL HBR
Common Name English
RIMITEROL HBR
Common Name English
Classification Tree Code System Code
NCI_THESAURUS C48149
Created by admin on Fri Dec 15 15:14:42 GMT 2023 , Edited by admin on Fri Dec 15 15:14:42 GMT 2023
Code System Code Type Description
ECHA (EC/EINECS)
250-834-6
Created by admin on Fri Dec 15 15:14:42 GMT 2023 , Edited by admin on Fri Dec 15 15:14:42 GMT 2023
PRIMARY
FDA UNII
I29DRR8S3R
Created by admin on Fri Dec 15 15:14:42 GMT 2023 , Edited by admin on Fri Dec 15 15:14:42 GMT 2023
PRIMARY
EPA CompTox
DTXSID70953756
Created by admin on Fri Dec 15 15:14:42 GMT 2023 , Edited by admin on Fri Dec 15 15:14:42 GMT 2023
PRIMARY
CAS
31842-61-2
Created by admin on Fri Dec 15 15:14:42 GMT 2023 , Edited by admin on Fri Dec 15 15:14:42 GMT 2023
PRIMARY
ChEMBL
CHEMBL1097630
Created by admin on Fri Dec 15 15:14:42 GMT 2023 , Edited by admin on Fri Dec 15 15:14:42 GMT 2023
PRIMARY
PUBCHEM
70685132
Created by admin on Fri Dec 15 15:14:42 GMT 2023 , Edited by admin on Fri Dec 15 15:14:42 GMT 2023
PRIMARY
NSC
289336
Created by admin on Fri Dec 15 15:14:42 GMT 2023 , Edited by admin on Fri Dec 15 15:14:42 GMT 2023
PRIMARY
MERCK INDEX
m9623
Created by admin on Fri Dec 15 15:14:42 GMT 2023 , Edited by admin on Fri Dec 15 15:14:42 GMT 2023
PRIMARY Merck Index
EVMPD
SUB04251MIG
Created by admin on Fri Dec 15 15:14:42 GMT 2023 , Edited by admin on Fri Dec 15 15:14:42 GMT 2023
PRIMARY
NCI_THESAURUS
C81646
Created by admin on Fri Dec 15 15:14:42 GMT 2023 , Edited by admin on Fri Dec 15 15:14:42 GMT 2023
PRIMARY
RXCUI
203161
Created by admin on Fri Dec 15 15:14:42 GMT 2023 , Edited by admin on Fri Dec 15 15:14:42 GMT 2023
PRIMARY RxNorm
SMS_ID
100000084921
Created by admin on Fri Dec 15 15:14:42 GMT 2023 , Edited by admin on Fri Dec 15 15:14:42 GMT 2023
PRIMARY