Piperolactam A

COC1=CC2=C3C(NC2=O)=CC4=CC=CC=C4C3=C1O

InChIKey=KBGNBPGXVKPRQI-UHFFFAOYSA-N

InChI=1S/C16H11NO3/c1-20-12-7-10-13-11(17-16(10)19)6-8-4-2-3-5-9(8)14(13)15(12)18/h2-7,18H,1H3,(H,17,19)

Targets

Primary Target	Pharmacology	Condition	Potency
Progesterone receptor 61 Target ID: P06401 Gene ID: 5241.0 Gene Symbol: PGR Target Organism: Homo sapiens (Human) Sources: https://www.ncbi.nlm.nih.gov/pubmed/28160639	Binding Agent 1064		0.249 µM [Ki]
Estrogen receptor 75 Target ID: P03372 Gene ID: 2099.0 Gene Symbol: ESR1 Target Organism: Homo sapiens (Human) Sources: https://www.ncbi.nlm.nih.gov/pubmed/28160639	Binding Agent 1064		0.294 µM [Ki]

PubMed

Title	Date	PubMed

Name

Type

Language

Piperolactam A

Common Name

English

1-Hydroxy-2-methoxydibenz[cd,f]indol-4(5H)-one

Systematic Name

English

Dibenz[cd,f]indol-4(5H)-one, 1-hydroxy-2-methoxy-

Systematic Name

English

14-Methoxy-15-oxidanyl-10-azatetracyclo(7.6.1.02,7.012,16)hexadeca-1(15),2,4,6,8,12(16),13-heptaen-11-one

Systematic Name

English

Code System Code Type Description

CAS

112501-42-5