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Details

Stereochemistry ACHIRAL
Molecular Formula C12H14N4O3S
Molecular Weight 294.33
Optical Activity NONE
Defined Stereocenters 0 / 0
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of SULFAMETOMIDINE

SMILES

COC1=CC(NS(=O)(=O)C2=CC=C(N)C=C2)=NC(C)=N1

InChI

InChIKey=QKLSCPPJEVXONT-UHFFFAOYSA-N
InChI=1S/C12H14N4O3S/c1-8-14-11(7-12(15-8)19-2)16-20(17,18)10-5-3-9(13)4-6-10/h3-7H,13H2,1-2H3,(H,14,15,16)

HIDE SMILES / InChI

Description

Sulfametomidine (or sulfamethomidine) is a sulfonamide antibacterial with a broad spectrum of activity; it’s an inhibitor of dihydrofolate reductase.

Approval Year

Unknown
139,594

Targets

Primary TargetPharmacologyConditionPotency
Bacterial dihydrofolate reductase
5
Inhibitor
8,297

Conditions

ConditionModalityTargetsHighest PhaseProduct
Bacterial infections
234
 Curative
Approved
8,429
METHOFADIN INJECTION

PubMed

Patents

US20140296310
1

Sample Use Guides

In Vivo Use Guide
initially 2 mg. subsequently 24 hour intervals in an average total dose of 6.3 mg.
Route of Administration: Other
In Vitro Use Guide
Unknown
ACTIVE MOIETY
Structure of SULFAMETOMIDINE
NIH
NCATS
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