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Details

Stereochemistry RACEMIC
Molecular Formula C10H15N.ClH
Molecular Weight 185.694
Optical Activity ( + / - )
Defined Stereocenters 0 / 1
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of PHENPROMETHAMINE HYDROCHLORIDE

SMILES

Cl.CNCC(C)C1=CC=CC=C1

InChI

InChIKey=OQHDRLTXPGYYJN-UHFFFAOYSA-N
InChI=1S/C10H15N.ClH/c1-9(8-11-2)10-6-4-3-5-7-10;/h3-7,9,11H,8H2,1-2H3;1H

HIDE SMILES / InChI

Description

Phenpromethamine is an adrenergic agent. Phenpromethamine was used as vasodilator agent. It is a stimulant which is banned in sport. It is available in supplements which are sold as fat burners or pre-workout boosters. Phenpromethamine is a potent CYP2D6 inhibitor.

Approval Year

1943
64

Overview

CYP3A4CYP2C9CYP2D6hERG
inhibitor
1,587
inhibitor
1,852

OverviewOther

Other InhibitorOther SubstrateOther Inducer

Drug as perpetrator​

PubMed

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