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Showing 1 - 2 of 2 results

Status:
Investigational

Class (Stereo):
CHEMICAL (ABSOLUTE)


Tirabrutinib (also known as ONO-4059 or GS-4059), a second-generation, enhanced-selectivity Bruton's tyrosine kinase inhibitor that demonstrated antitumor activity in preclinical models. Tirabrutinib participated in phase I clinical trial in patients...
Status:
Investigational

Class (Stereo):
CHEMICAL (ACHIRAL)


PQR-309 is an orally bioavailable pan inhibitor of phosphoinositide-3-kinases (PI3K) and inhibitor of the mammalian target of rapamycin (mTOR), with potential antineoplastic activity. PI3K/mTOR kinase inhibitor PQR-309 inhibits the PI3K kinase isofor...