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Showing 1 - 6 of 6 results

Status:
US Approved Rx (2007)
First approved in 2007

Class (Stereo):
CHEMICAL (ACHIRAL)



Nilotinib (AMN107, trade name Tasigna) is a kinase inhibitor indicated for the treatment of chronic phase and accelerated phase Philadelphia chromosome-positive chronic myelogenous leukemia (CML) in adult patients resistant to or intolerant to prior ...
Status:
Investigational

Class (Stereo):
CHEMICAL (ABSOLUTE)



Tanespimycin (17-allylamino-17-demethoxygeldanamycin, 17-AAG) is a synthetic analogue of geldanamycin, an antibiotic first purified in 1970 from Streptomyces hygroscopicus. Tanespimycin is an Hsp90 inhibitor that has demonstrated the potential to dis...
Status:
Designated

Class (Stereo):
CHEMICAL (ACHIRAL)

NRC-AN-019 has been found to be a promising new lead compound for the therapy of imatinib mesylate-resistant chronic myeloid leukemia. NRC-AN-019 showed considerable safety and response. In addition, it has the therapeutic potential in the treatment ...
Status:
US Approved Rx (2002)
First approved in 2002

Class:
PROTEIN

Status:
Investigational

Class:
PROTEIN

Status:
US Approved Rx (2025)
First approved in 2006

Class (Stereo):
CHEMICAL (ACHIRAL)



Dasatinib [BMS 354825] is an orally active, small molecule, dual inhibitor of both SRC and ABL kinases that is under development with Bristol-Myers Squibb for the treatment of patients with chronic myelogenous leukaemia (CML) and imatinib-acquired re...