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Development Status

US Approved Rx

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Primary Target

Kappa opioid receptor

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Mu opioid receptor

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Highest Phase

Approved

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Approval Year

1967

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Condition

Pain

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Primary

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CNS Activity

CNS Active

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Originator

Tullar, B.F.|Harris, L.S.|Perry, R.L.|Pierson, A.K.|Soria, A.E.|Wetterau, W.F.|Albertson, N.F.

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OPIOIDS

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ATC Level 4

Benzomorphan derivatives

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Salts, Hydrates, Esters, etc.

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Showing 1 - 4 of 4 results

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PENTAZOCINE

RP4A60D26L

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Status:

US Approved Rx (1997)

First approved in 1967

Class (Stereo):

CHEMICAL (RACEMIC)

Targets:

Mu opioid receptor

Kappa opioid receptor

Conditions:

Pentazocine is a synthetically prepared prototypical mixed agonist-antagonist narcotic (opioid analgesic) drug of the benzomorphan class of opioids used to treat moderate to moderately severe pain. Pentazocine is sold under several brand names, such ...

as Fortral, Sosegon, Talwin NX. Pentazocine acts as an agonist of κ-opioid receptors and as an antagonist of μ-opioid receptors. This compound may exist as one of two enantiomers, named (+)-pentazocine and (−)-pentazocine. Side effects are similar to those of morphine, but pentazocine, due to its action at the kappa opioid receptor is more likely to invoke psychotomimetic effects. High dose may cause high blood pressure or high heart rate.

PENTAZOCINE HYDROCHLORIDE

A36BXO4PPX

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Status:

US Approved Rx (1997)

First approved in 1967

Class (Stereo):

CHEMICAL (RACEMIC)

Targets:

Mu opioid receptor

Kappa opioid receptor

Conditions:

Pentazocine is a synthetically prepared prototypical mixed agonist-antagonist narcotic (opioid analgesic) drug of the benzomorphan class of opioids used to treat moderate to moderately severe pain. Pentazocine is sold under several brand names, such ...

as Fortral, Sosegon, Talwin NX. Pentazocine acts as an agonist of κ-opioid receptors and as an antagonist of μ-opioid receptors. This compound may exist as one of two enantiomers, named (+)-pentazocine and (−)-pentazocine. Side effects are similar to those of morphine, but pentazocine, due to its action at the kappa opioid receptor is more likely to invoke psychotomimetic effects. High dose may cause high blood pressure or high heart rate.

PENTAZOCINE LACTATE

1P2XIB510O

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Status:

US Approved Rx (1997)

First approved in 1967

Class (Stereo):

CHEMICAL (MIXED)

Targets:

Mu opioid receptor

Kappa opioid receptor

Conditions:

Pentazocine is a synthetically prepared prototypical mixed agonist-antagonist narcotic (opioid analgesic) drug of the benzomorphan class of opioids used to treat moderate to moderately severe pain. Pentazocine is sold under several brand names, such ...

as Fortral, Sosegon, Talwin NX. Pentazocine acts as an agonist of κ-opioid receptors and as an antagonist of μ-opioid receptors. This compound may exist as one of two enantiomers, named (+)-pentazocine and (−)-pentazocine. Side effects are similar to those of morphine, but pentazocine, due to its action at the kappa opioid receptor is more likely to invoke psychotomimetic effects. High dose may cause high blood pressure or high heart rate.

PENTAZOCINE, (-)-

768DQ5A5AI

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Status:

US Approved Rx (1997)

First approved in 1967

Class (Stereo):

CHEMICAL (ABSOLUTE)

Targets:

Mu opioid receptor

Kappa opioid receptor

Conditions:

Pentazocine is a synthetically prepared prototypical mixed agonist-antagonist narcotic (opioid analgesic) drug of the benzomorphan class of opioids used to treat moderate to moderately severe pain. Pentazocine is sold under several brand names, such ...

as Fortral, Sosegon, Talwin NX. Pentazocine acts as an agonist of κ-opioid receptors and as an antagonist of μ-opioid receptors. This compound may exist as one of two enantiomers, named (+)-pentazocine and (−)-pentazocine. Side effects are similar to those of morphine, but pentazocine, due to its action at the kappa opioid receptor is more likely to invoke psychotomimetic effects. High dose may cause high blood pressure or high heart rate.

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