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Showing 1 - 5 of 5 results

Status:
Investigational

Class (Stereo):
CHEMICAL (ABSOLUTE)



Nastorazepide (Z-360) is a selective, orally available, gastrin/cholecystokinin 2 (CCK-2) receptor antagonist with potential antineoplastic activity. Z-360 binds to the gastrin/CCK-2 receptor, thereby preventing receptor activation by gastrin, a pept...
Status:
Investigational

Class (Stereo):
CHEMICAL (ACHIRAL)



Rigosertib sodium (ON 01910.Na) is a small molecule inhibitor of critical pathways important in the growth and survival of cancer cells, being developed by Onconova Therapeutics ("Onconova") for the treatment of hematologic malignancies and solid tum...
Status:
Investigational

Class (Stereo):
CHEMICAL (ABSOLUTE)



RO4929097 (R-4733) is a small-molecule inhibitor of gamma-secretase (γ-secretase) with high oral bioavailability leading to the blockade of Notch signaling in tumor cells. This compound was co-developed by Roche and National Cancer Institute (NCI). ...
Status:
Investigational

Class (Stereo):
CHEMICAL (ABSOLUTE)



Nastorazepide (Z-360) is a selective, orally available, gastrin/cholecystokinin 2 (CCK-2) receptor antagonist with potential antineoplastic activity. Z-360 binds to the gastrin/CCK-2 receptor, thereby preventing receptor activation by gastrin, a pept...
Status:
Investigational

Class (Stereo):
CHEMICAL (ACHIRAL)



Rigosertib sodium (ON 01910.Na) is a small molecule inhibitor of critical pathways important in the growth and survival of cancer cells, being developed by Onconova Therapeutics ("Onconova") for the treatment of hematologic malignancies and solid tum...