Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 21:52:29 GMT 2025
by
admin
on
Tue Apr 01 21:52:29 GMT 2025
|
| Protein Type | RECEPTOR |
| Protein Sub Type | Other |
| Sequence Origin | HUMAN |
| Sequence Type | COMPLETE |
| Record UNII |
ZFQG2GI3F2
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| Record Status |
Validated (UNII)
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| Record Version |
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-
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Preferred Name | English | ||
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| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
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301156-53-6
Created by
admin on Tue Apr 01 21:52:29 GMT 2025 , Edited by admin on Tue Apr 01 21:52:29 GMT 2025
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PRIMARY | |||
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ZFQG2GI3F2
Created by
admin on Tue Apr 01 21:52:29 GMT 2025 , Edited by admin on Tue Apr 01 21:52:29 GMT 2025
|
PRIMARY | |||
|
Q06124
Created by
admin on Tue Apr 01 21:52:29 GMT 2025 , Edited by admin on Tue Apr 01 21:52:29 GMT 2025
|
PRIMARY |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
ALLOSTERIC INHIBITOR->TARGET |
IN-VITRO
IC50
|
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ACTIVATOR->OFF TARGET |
Kd
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
ALLOSTERIC INHIBITOR
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INHIBITOR -> TARGET |
Greatly reduced effect in the SHP2 E76K or T253M/Q257L mutants.
ALLOSTERIC
IC50
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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Structural Modifications
| Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
|---|---|---|---|---|---|---|
| AMINO_ACID_SUBSTITUTION | [1_1] | N-TERMINUS | N-ACETYLTHREONINE | V0E98V3R9O | ||
| AMINO_ACID_SUBSTITUTION | [1_61] [1_65] [1_545] [1_583] | SITE_SPECIFIC | TYROSINE O-PHOSPHATE | 2R86C98KDX |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT:NUMBER(CALCULATED) | CHEMICAL |
|