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Approval Year

Substance Class Protein
Created
by admin
on Sat Dec 16 14:38:13 UTC 2023
Edited
by admin
on Sat Dec 16 14:38:13 UTC 2023
Protein Sub Type ION CHANNEL
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
ZEX6X6B5QP
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
AMILORIDE-SENSITIVE SODIUM CHANNEL
Common Name English
Epithelial Sodium Channel–
Common Name English
ENAC
Common Name English
Epithelial Na(+) channel
Common Name English
Nonvoltage-gated sodium channel 1
Common Name English
Code System Code Type Description
UNIPROT
P51168
Created by admin on Sat Dec 16 14:38:13 UTC 2023 , Edited by admin on Sat Dec 16 14:38:13 UTC 2023
PRIMARY
UNIPROT
P37088
Created by admin on Sat Dec 16 14:38:13 UTC 2023 , Edited by admin on Sat Dec 16 14:38:13 UTC 2023
PRIMARY
UNIPROT
P51170
Created by admin on Sat Dec 16 14:38:13 UTC 2023 , Edited by admin on Sat Dec 16 14:38:13 UTC 2023
PRIMARY
FDA UNII
ZEX6X6B5QP
Created by admin on Sat Dec 16 14:38:13 UTC 2023 , Edited by admin on Sat Dec 16 14:38:13 UTC 2023
PRIMARY
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 2_260
N 3_209
N 3_497
Related Record Type Details
INHIBITOR -> TARGET
Binds selectively to ENaC and promotes internalization of the a-, b-, and g-subunits. Removing ENaC from the membrane with SPX-101 causes a significant decrease in amiloride-sensitive current.
EC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL
Molecular Formula CHEMICAL