U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 16:56:30 GMT 2025
Edited
by admin
on Tue Apr 01 16:56:30 GMT 2025
Protein Sub Type
Sequence Type COMPLETE
Record UNII
Z789E7KP9Q
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
MAP KINASE SIGNAL-INTEGRATING KINASE 1
Preferred Name English
MAP KINASE-INTERACTING SERINE/THREONINE-PROTEIN KINASE 1
Common Name English
MAPK SIGNAL-INTEGRATING KINASE 1
Common Name English
MNK1
Common Name English
MKNK1
Common Name English
Code System Code Type Description
WIKIPEDIA
MKNK1
Created by admin on Tue Apr 01 16:56:30 GMT 2025 , Edited by admin on Tue Apr 01 16:56:30 GMT 2025
PRIMARY
UNIPROT
Q9BUB5
Created by admin on Tue Apr 01 16:56:30 GMT 2025 , Edited by admin on Tue Apr 01 16:56:30 GMT 2025
PRIMARY
FDA UNII
Z789E7KP9Q
Created by admin on Tue Apr 01 16:56:30 GMT 2025 , Edited by admin on Tue Apr 01 16:56:30 GMT 2025
PRIMARY
PHAROS
Q9BUB5
Created by admin on Tue Apr 01 16:56:30 GMT 2025 , Edited by admin on Tue Apr 01 16:56:30 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_39] [1_221] [1_226] [1_460] S DEXFOSFOSERINE VI4F0K069V
AMINO ACID SUBSTITUTION [1_250] [1_255] T THREONINE PHOSPHATE 3L4WX7B1EI
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL