U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Mon Mar 31 22:55:32 GMT 2025
Edited
by admin
on Mon Mar 31 22:55:32 GMT 2025
Protein Type MONOCLONAL ANTIBODY
Protein Sub Type IGG1
Sequence Origin HUMANIZED MOUSE
Sequence Type COMPLETE
Record UNII
Y6M3205516
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
lumretuzumab [INN]
Preferred Name English
LUMRETUZUMAB
INN   USAN   WHO-DD  
INN   USAN  
Official Name English
RO-5479599
Code English
Lumretuzumab [WHO-DD]
Common Name English
RG7116
Code English
RG-7116
Code English
RO5479599
Code English
IMMUNOGLOBULIN G1-KAPPA, ANTI-(HOMO SAPIENS ERBB3 (RECEPTOR TYROSINE-PROTEIN KINASE ERBB-3, HER3)), HUMANIZED MONOCLONAL ANTIBODY
Common Name English
LUMRETUZUMAB [USAN]
Common Name English
Code System Code Type Description
USAN
CD-100
Created by admin on Mon Mar 31 22:55:32 GMT 2025 , Edited by admin on Mon Mar 31 22:55:32 GMT 2025
PRIMARY
ChEMBL
CHEMBL3707404
Created by admin on Mon Mar 31 22:55:32 GMT 2025 , Edited by admin on Mon Mar 31 22:55:32 GMT 2025
PRIMARY
WIKIPEDIA
Lumretuzumab
Created by admin on Mon Mar 31 22:55:32 GMT 2025 , Edited by admin on Mon Mar 31 22:55:32 GMT 2025
PRIMARY
EVMPD
SUB177214
Created by admin on Mon Mar 31 22:55:32 GMT 2025 , Edited by admin on Mon Mar 31 22:55:32 GMT 2025
PRIMARY
DRUG BANK
DB12683
Created by admin on Mon Mar 31 22:55:32 GMT 2025 , Edited by admin on Mon Mar 31 22:55:32 GMT 2025
PRIMARY
FDA UNII
Y6M3205516
Created by admin on Mon Mar 31 22:55:32 GMT 2025 , Edited by admin on Mon Mar 31 22:55:32 GMT 2025
PRIMARY
SMS_ID
100000163088
Created by admin on Mon Mar 31 22:55:32 GMT 2025 , Edited by admin on Mon Mar 31 22:55:32 GMT 2025
PRIMARY
ChEMBL
CHEMBL2109441
Created by admin on Mon Mar 31 22:55:32 GMT 2025 , Edited by admin on Mon Mar 31 22:55:32 GMT 2025
PRIMARY
INN
9952
Created by admin on Mon Mar 31 22:55:32 GMT 2025 , Edited by admin on Mon Mar 31 22:55:32 GMT 2025
PRIMARY
CAS
1448327-63-6
Created by admin on Mon Mar 31 22:55:32 GMT 2025 , Edited by admin on Mon Mar 31 22:55:32 GMT 2025
PRIMARY
NCI_THESAURUS
C104058
Created by admin on Mon Mar 31 22:55:32 GMT 2025 , Edited by admin on Mon Mar 31 22:55:32 GMT 2025
PRIMARY
From To
1_22 1_96
1_147 1_203
1_264 1_324
1_370 1_428
2_22 2_96
2_147 2_203
2_264 2_324
2_370 2_428
3_23 3_94
3_140 3_200
4_23 4_94
4_140 4_200
1_223 3_220
2_223 4_220
1_229 2_229
1_232 2_232
Glycosylation Link Type Site
N 1_300
N 2_300
Related Record Type Details
TARGET -> INHIBITOR
Related Record Type Details
ACTIVE MOIETY

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO_ACID_SUBSTITUTION [1_1] [2_1] 5'-TERMINUS PIDOLIC ACID SZB83O1W42
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL
Molecular Formula CHEMICAL