Approval Year
Substance Class |
Protein
Created
by
admin
on
Edited
Sat Dec 16 11:42:57 GMT 2023
by
admin
on
Sat Dec 16 11:42:57 GMT 2023
|
Protein Sub Type | |
Sequence Type | COMPLETE |
Record UNII |
Y154T023U0
|
Record Status |
Validated (UNII)
|
Record Version |
|
-
Download
Name | Type | Language | ||
---|---|---|---|---|
|
Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English |
Code System | Code | Type | Description | ||
---|---|---|---|---|---|
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Y154T023U0
Created by
admin on Sat Dec 16 11:43:00 GMT 2023 , Edited by admin on Sat Dec 16 11:43:00 GMT 2023
|
PRIMARY | |||
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P29274
Created by
admin on Sat Dec 16 11:43:00 GMT 2023 , Edited by admin on Sat Dec 16 11:43:00 GMT 2023
|
PRIMARY | |||
|
P29274
Created by
admin on Sat Dec 16 11:43:00 GMT 2023 , Edited by admin on Sat Dec 16 11:43:00 GMT 2023
|
PRIMARY |
From | To |
---|---|
1_71 | 1_159 |
1_74 | 1_146 |
1_77 | 1_166 |
1_259 | 1_262 |
Glycosylation Type | HUMAN |
Glycosylation Link Type | Site |
---|---|
N | 1_154 |
Related Record | Type | Details | ||
---|---|---|---|---|
|
AGONIST -> TARGET |
BINDING
Kd
|
||
|
INHIBITOR -> TARGET | |||
|
AGONIST -> TARGET |
|
||
|
INHIBITOR -> TARGET |
BINDING
IC50
|
||
|
AGONIST -> TARGET |
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET | |||
|
AGONIST -> TARGET |
|
||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
Approximately 1000-fold more selective
over other ARs.
Ki
|
||
|
INHIBITOR -> TARGET |
Ki
|
||
|
INHIBITOR -> TARGET |
Highly selective over hA2B Ki = 1110 nM.
Ki
|
||
|
INHIBITOR -> TARGET |
ANTAGONIST
IC50
|
||
|
RADIOLIGAND->TARGET |
|
||
|
INHIBITOR -> TARGET |
ANTAGONIST
Ki
|
||
|
AGONIST -> TARGET |
BINDING
IC50
|
||
|
RADIOLIGAND->TARGET |
BINDING
Kd
|
||
|
INHIBITOR -> TARGET |
Ki
|
||
|
WEAK AGONIST->OFF TARGET |
Rat brain receptor
BINDING
Ki
|
||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
|
||
|
RADIOLIGAND->TARGET |
Ki
|
||
|
INHIBITOR -> TARGET |
BINDING
IC50
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET |
|
||
|
INHIBITOR -> TARGET |
selective antagonsist
Ki
|
||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
BINDING
IC50
|
||
|
INHIBITOR -> TARGET |
Showed high selectivity over other adenosine receptors.
Ki
|
||
|
WEAK INHIBITOR->TARGET |
Nonselective adenosine receptor antagonist. May be responsible for pain relief.
Ki
|
||
|
AGONIST -> TARGET |
|
||
|
INHIBITOR -> TARGET |
Kb actually
Kd
|
||
|
RADIOLIGAND->TARGET |
Kd
|
||
|
AGONIST -> TARGET |
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INVERSE AGONIST->TARGET |
EC50
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INHIBITOR -> TARGET |
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|
INHIBITOR -> TARGET |
IC50
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||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
ANTAGONIST
Ki
|
||
|
AGONIST -> TARGET |
|
Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
---|---|---|---|---|---|---|
Molecular Formula | CHEMICAL |
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||||
MOL_WEIGHT | CHEMICAL |
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