U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Wed Apr 02 07:19:50 GMT 2025
Edited
by admin
on Wed Apr 02 07:19:50 GMT 2025
Protein Type MONOCLONAL ANTIBODY
Protein Sub Type IGG1
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
XI9R476VH8
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
idactamab [INN]
Preferred Name English
IDACTAMAB
INN  
Official Name English
IMMUNOGLOBULIN G1 (243A-CYSTEINE), ANTI-(HUMAN AMINO ACID TRANSPORTER ASCT2) (HUMAN MONOCLONAL INT-001 .GAMMA.1-CHAIN), DISULFIDE WITH HUMAN MONOCLONAL INT-001 .KAPPA.-CHAIN, DIMER
Common Name English
Code System Code Type Description
INN
11348
Created by admin on Wed Apr 02 07:19:50 GMT 2025 , Edited by admin on Wed Apr 02 07:19:50 GMT 2025
PRIMARY
NCI_THESAURUS
C175797
Created by admin on Wed Apr 02 07:19:50 GMT 2025 , Edited by admin on Wed Apr 02 07:19:50 GMT 2025
PRIMARY
FDA UNII
XI9R476VH8
Created by admin on Wed Apr 02 07:19:50 GMT 2025 , Edited by admin on Wed Apr 02 07:19:50 GMT 2025
PRIMARY
CAS
2245205-37-0
Created by admin on Wed Apr 02 07:19:50 GMT 2025 , Edited by admin on Wed Apr 02 07:19:50 GMT 2025
PRIMARY
SMS_ID
300000035006
Created by admin on Wed Apr 02 07:19:50 GMT 2025 , Edited by admin on Wed Apr 02 07:19:50 GMT 2025
PRIMARY
From To
4_134 4_194
3_134 3_194
2_266 2_326
2_224 4_214
2_148 2_204
2_22 2_95
1_372 1_430
1_266 1_326
1_224 3_214
1_233 2_233
1_230 2_230
1_22 1_95
1_148 1_204
2_372 2_430
3_23 3_88
4_23 4_88
Glycosylation Type MAMMALIAN
Glycosylation Link Type Site
N 1_302
N 2_302
Related Record Type Details
ACTIVE MOIETY
Immunomodulator, antineoplastic

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO_ACID_SUBSTITUTION [1_1] [2_1] N-TERMINUS PIDOLIC ACID SZB83O1W42
AMINO ACID REMOVAL [1_452] [2_452] C-TERMINUS LYSINE K3Z4F929H6
Name Property Type Amount Referenced Substance Defining Parameters References
Molecular Formula CHEMICAL
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL