U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Wed Apr 02 12:27:38 GMT 2025
Edited
by admin
on Wed Apr 02 12:27:38 GMT 2025
Protein Type MONOCLONAL ANTIBODY CONJUGATE
Protein Sub Type IGG1|KAPPA
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
VG5Y3A9DFS
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
H-gamma1 heavy chain Homo sapiens (1-450) [VH (Homo sapiens IGHV4-39*01 (96.0%) -(IGHD) -IGHJ5*02 (93.8%), CDR-IMGT [10.7.12] (26-35.53-59.98-109)) (1-120) -Homo sapiens IGHG1*01 (100%) G1m17,1 CH1 K120, CH3 D12, L14 (CH1 K120 (217) (121-218), hinge 1-15
Preferred Name English
Felmetatug Vedotin
INN  
Official Name English
Immunoglobulin G1, anti-(human/Macaca fascicularis/Mus musculus B7 homolog protein B7H4) (human monoclonal B7H41001 ?1-chain), disulfide with human monoclonal B7H41001 ?-chain, dimer, reduced, tetrakis(thioether) with N-[[[4-[[N-[6-(3-mercapto-2,5-dioxo-
Common Name English
immunoglobulin G1-kappa, anti-[Homo sapiens VTCN1 (V-set domain containing T cell activation inhibitor 1, B7 family member H4, B7H4, B7-H4)], Homo sapiens monoclonal antibody, conjugated on an average of four cysteinyl residues to vedotin, comprising a c
Common Name English
felmetatug vedotin [INN]
Common Name English
Code System Code Type Description
CAS
2924808-30-8
Created by admin on Wed Apr 02 12:27:38 GMT 2025 , Edited by admin on Wed Apr 02 12:27:38 GMT 2025
PRIMARY
SMS_ID
300000039890
Created by admin on Wed Apr 02 12:27:38 GMT 2025 , Edited by admin on Wed Apr 02 12:27:38 GMT 2025
PRIMARY
FDA UNII
VG5Y3A9DFS
Created by admin on Wed Apr 02 12:27:38 GMT 2025 , Edited by admin on Wed Apr 02 12:27:38 GMT 2025
PRIMARY
NCI_THESAURUS
C186669
Created by admin on Wed Apr 02 12:27:38 GMT 2025 , Edited by admin on Wed Apr 02 12:27:38 GMT 2025
PRIMARY
INN
13231
Created by admin on Wed Apr 02 12:27:38 GMT 2025 , Edited by admin on Wed Apr 02 12:27:38 GMT 2025
PRIMARY
From To
1_22 1_97
2_22 2_97
2_147 2_203
2_223 4_214
2_264 2_324
1_147 1_203
2_370 2_428
3_23 3_88
3_134 3_194
4_23 4_88
4_134 4_194
1_223 3_214
1_229 2_229
1_232 2_232
1_264 1_324
1_370 1_428
Glycosylation Type MAMMALIAN
Glycosylation Link Type Site
N 1_300
N 2_300
Related Record Type Details
PARENT -> CONJUGATE
TARGET -> INHIBITOR
PRECLINICAL
TOXIN -> CONJUGATE
Related Record Type Details
ACTIVE MOIETY
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL