U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 18:26:54 GMT 2025
Edited
by admin
on Tue Apr 01 18:26:54 GMT 2025
Protein Sub Type
Sequence Type COMPLETE
Record UNII
UYB9SX45Y8
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
CAMP-SPECIFIC 3',5'-CYCLIC PHOSPHODIESTERASE 7B
Common Name English
PDE7B
Preferred Name English
Code System Code Type Description
FDA UNII
UYB9SX45Y8
Created by admin on Tue Apr 01 18:26:54 GMT 2025 , Edited by admin on Tue Apr 01 18:26:54 GMT 2025
PRIMARY
UNIPROT
Q9NP56
Created by admin on Tue Apr 01 18:26:54 GMT 2025 , Edited by admin on Tue Apr 01 18:26:54 GMT 2025
PRIMARY
PHAROS
Q9NP56
Created by admin on Tue Apr 01 18:26:54 GMT 2025 , Edited by admin on Tue Apr 01 18:26:54 GMT 2025
PRIMARY
Related Record Type Details
RADIOLIGAND->TARGET
Selective PDE7 inhibitor. Percent inhibition of other PDEs (PDE1A, 3A, 5A, 6, 8A1, 9A2, and 11A4) by 1 ?M of MTP38 were less than 50%.
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
Selective PDE7 inhibitor. Percent inhibition of other PDEs (PDE1A, 3A, 5A, 6, 8A1, 9A2, and 11A4) by 1 ?M of MTP38 were less than 50%.
IC50

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_426] DEXFOSFOSERINE VI4F0K069V
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL