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Details

Stereochemistry ACHIRAL
Molecular Formula C21H27NO2
Molecular Weight 325.4446
Optical Activity NONE
Defined Stereocenters 0 / 0
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of DIETIFEN

SMILES

CCN(CC)CCOC1=CC=C(C=C1)C(=O)CCC2=CC=CC=C2

InChI

InChIKey=KMICWMXRUOETFR-UHFFFAOYSA-N
InChI=1S/C21H27NO2/c1-3-22(4-2)16-17-24-20-13-11-19(12-14-20)21(23)15-10-18-8-6-5-7-9-18/h5-9,11-14H,3-4,10,15-17H2,1-2H3

HIDE SMILES / InChI

Molecular Formula C21H27NO2
Molecular Weight 325.4446
Charge 0
Count
Stereochemistry ACHIRAL
Additional Stereochemistry No
Defined Stereocenters 0 / 0
E/Z Centers 0
Optical Activity NONE

Dietifen is an anesthetic, vasodilator and antifungal agent. The main pharmacological feature of the drug is its ability to cause expansion of the coronary vessels. It also has a moderate spasmolytic activity (reduces spasms of the muscles of the intestine and other internal organs) and somewhat inhibits the conduction of nervous excitement through the vegetative nodes. Significant changes in blood pressure and pulse rate does not cause, does not possess hormonal (estrogenic) activity. It is indicated for the treatment of chronic coronary insufficiency, angina pectoris, severe forms of coronary sclerosis and pre-infarction conditions (simultaneously with anticoagulants).

Approval Year

Targets

Targets

Primary TargetPharmacologyConditionPotency
Patents

Sample Use Guides

In Vivo Use Guide
25 mg 3-4 times a day (after meals). Treatment is carried out by courses for 2-3 weeks.
Route of Administration: Oral
Substance Class Chemical
Created
by admin
on Fri Dec 15 16:25:15 GMT 2023
Edited
by admin
on Fri Dec 15 16:25:15 GMT 2023
Record UNII
UO003HH66V
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
DIETIFEN
INN  
INN  
Official Name English
dietifen [INN]
Common Name English
EPILIN
Common Name English
4-(2-(DIETHYLAMINO)ETHOXY)PHENYL PHENETHYL KETONE
Systematic Name English
Classification Tree Code System Code
NCI_THESAURUS C514
Created by admin on Fri Dec 15 16:25:15 GMT 2023 , Edited by admin on Fri Dec 15 16:25:15 GMT 2023
Code System Code Type Description
SMS_ID
100000083150
Created by admin on Fri Dec 15 16:25:15 GMT 2023 , Edited by admin on Fri Dec 15 16:25:15 GMT 2023
PRIMARY
FDA UNII
UO003HH66V
Created by admin on Fri Dec 15 16:25:15 GMT 2023 , Edited by admin on Fri Dec 15 16:25:15 GMT 2023
PRIMARY
EVMPD
SUB07115MIG
Created by admin on Fri Dec 15 16:25:15 GMT 2023 , Edited by admin on Fri Dec 15 16:25:15 GMT 2023
PRIMARY
ChEMBL
CHEMBL2104343
Created by admin on Fri Dec 15 16:25:15 GMT 2023 , Edited by admin on Fri Dec 15 16:25:15 GMT 2023
PRIMARY
EPA CompTox
DTXSID90190348
Created by admin on Fri Dec 15 16:25:15 GMT 2023 , Edited by admin on Fri Dec 15 16:25:15 GMT 2023
PRIMARY
INN
2794
Created by admin on Fri Dec 15 16:25:15 GMT 2023 , Edited by admin on Fri Dec 15 16:25:15 GMT 2023
PRIMARY
NCI_THESAURUS
C78039
Created by admin on Fri Dec 15 16:25:15 GMT 2023 , Edited by admin on Fri Dec 15 16:25:15 GMT 2023
PRIMARY
PUBCHEM
208834
Created by admin on Fri Dec 15 16:25:15 GMT 2023 , Edited by admin on Fri Dec 15 16:25:15 GMT 2023
PRIMARY
CAS
3686-78-0
Created by admin on Fri Dec 15 16:25:15 GMT 2023 , Edited by admin on Fri Dec 15 16:25:15 GMT 2023
PRIMARY
Related Record Type Details
ACTIVE MOIETY