U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS
This repository is under review for potential modification in compliance with Administration directives.

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 18:25:47 GMT 2025
Edited
by admin
on Tue Apr 01 18:25:47 GMT 2025
Protein Sub Type
Sequence Type COMPLETE
Record UNII
TFZ3H25BS1
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
AMPA-SELECTIVE GLUTAMATE RECEPTOR 1
Preferred Name English
GLUTAMATE RECEPTOR 1
Common Name English
GLUR-K1
Common Name English
GLUTAMATE RECEPTOR IONOTROPIC, AMPA 1
Common Name English
GLUR-A
Common Name English
GLUH1
Common Name English
GLUR1
Common Name English
Code System Code Type Description
FDA UNII
TFZ3H25BS1
Created by admin on Tue Apr 01 18:25:47 GMT 2025 , Edited by admin on Tue Apr 01 18:25:47 GMT 2025
PRIMARY
UNIPROT
P42261
Created by admin on Tue Apr 01 18:25:47 GMT 2025 , Edited by admin on Tue Apr 01 18:25:47 GMT 2025
PRIMARY
From To
1_57 1_305
1_714 1_769
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_45
N 1_231
N 1_239
N 1_345
N 1_383
N 1_388
Related Record Type Details
ACTIVATOR -> TARGET
AMPA-R potentiator with little agonistic effect
ALLOSTERIC ACTIVATOR
INHIBITOR -> TARGET
ACTIVATOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
ACTIVATOR -> TARGET
AMPA Receptor potentiators
ALLOSTERIC ACTIVATOR
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_627] [1_692] [1_831] [1_845] DEXFOSFOSERINE VI4F0K069V
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL