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Details

Stereochemistry ACHIRAL
Molecular Formula C22H23ClFN5O2.2C7H8O3S
Molecular Weight 788.305
Optical Activity NONE
Defined Stereocenters 0 / 0
E/Z Centers 1
Charge 0

SHOW SMILES / InChI
Structure of NEPTINIB DITOSYLATE

SMILES

CC1=CC=C(C=C1)S(O)(=O)=O.CC2=CC=C(C=C2)S(O)(=O)=O.CCOC3=C(NC(=O)\C=C\CN(C)C)C=C4C(NC5=CC=C(F)C(Cl)=C5)=NC=NC4=C3

InChI

InChIKey=MCEGMGYYDQRIMH-TXOOBNKBSA-N
InChI=1S/C22H23ClFN5O2.2C7H8O3S/c1-4-31-20-12-18-15(11-19(20)28-21(30)6-5-9-29(2)3)22(26-13-25-18)27-14-7-8-17(24)16(23)10-14;2*1-6-2-4-7(5-3-6)11(8,9)10/h5-8,10-13H,4,9H2,1-3H3,(H,28,30)(H,25,26,27);2*2-5H,1H3,(H,8,9,10)/b6-5+;;

HIDE SMILES / InChI

Molecular Formula C7H8O3S
Molecular Weight 172.202
Charge 0
Count
Stereochemistry ACHIRAL
Additional Stereochemistry No
Defined Stereocenters 0 / 0
E/Z Centers 0
Optical Activity NONE

Molecular Formula C22H23ClFN5O2
Molecular Weight 443.902
Charge 0
Count
Stereochemistry ACHIRAL
Additional Stereochemistry No
Defined Stereocenters 0 / 0
E/Z Centers 1
Optical Activity NONE

Approval Year

Substance Class Chemical
Created
by admin
on Tue Apr 01 22:14:24 GMT 2025
Edited
by admin
on Tue Apr 01 22:14:24 GMT 2025
Record UNII
TA6UHD60QT
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
NEPTINIB DI-P-METHYLBENZENESULFONATE
Preferred Name English
NEPTINIB DITOSYLATE
Common Name English
2-BUTENAMIDE, N-(4-((3-CHLORO-4-FLUOROPHENYL)AMINO)-7-ETHOXY-6-QUINAZOLINYL)-4-(DIMETHYLAMINO)-, (2E)-, 4-METHYLBENZENESULFONATE (1:2)
Systematic Name English
2-BUTENAMIDE, N-(4-((3-CHLORO-4-FLUOROPHENYL)AMINO)-7-ETHOXY-6-QUINAZOLINYL)-4-(DIMETHYLAMINO)-, 4-METHYLBENZENESULFONATE (1:2)
Systematic Name English
Code System Code Type Description
CAS
2085843-54-3
Created by admin on Tue Apr 01 22:14:24 GMT 2025 , Edited by admin on Tue Apr 01 22:14:24 GMT 2025
PRIMARY
CAS
1957132-03-4
Created by admin on Tue Apr 01 22:14:24 GMT 2025 , Edited by admin on Tue Apr 01 22:14:24 GMT 2025
NON-SPECIFIC STEREOCHEMISTRY
PUBCHEM
132164922
Created by admin on Tue Apr 01 22:14:24 GMT 2025 , Edited by admin on Tue Apr 01 22:14:24 GMT 2025
PRIMARY
FDA UNII
TA6UHD60QT
Created by admin on Tue Apr 01 22:14:24 GMT 2025 , Edited by admin on Tue Apr 01 22:14:24 GMT 2025
PRIMARY
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