U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS
This repository is under review for potential modification in compliance with Administration directives.

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 23:42:39 GMT 2025
Edited
by admin
on Tue Apr 01 23:42:39 GMT 2025
Protein Type ENZYME
Protein Sub Type TYROSINE KINASE
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
S64UQ6O9VK
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
CD117 D816V
Preferred Name English
MAST/STEM CELL GROWTH FACTOR RECEPTOR KIT D816V
Common Name English
PIEBALD TRAIT PROTEIN D816V
Common Name English
TYROSINE-PROTEIN KINASE KIT D816V
Common Name English
V-KIT HARDY-ZUCKERMAN 4 FELINE SARCOMA VIRAL ONCOGENE HOMOLOG D816V
Common Name English
KIT D816V
Common Name English
SCFR D816V
Common Name English
Code System Code Type Description
UNIPROT
P10721
Created by admin on Tue Apr 01 23:42:39 GMT 2025 , Edited by admin on Tue Apr 01 23:42:39 GMT 2025
PRIMARY
FDA UNII
S64UQ6O9VK
Created by admin on Tue Apr 01 23:42:39 GMT 2025 , Edited by admin on Tue Apr 01 23:42:39 GMT 2025
PRIMARY
WIKIPEDIA
CD117
Created by admin on Tue Apr 01 23:42:39 GMT 2025 , Edited by admin on Tue Apr 01 23:42:39 GMT 2025
PRIMARY
EC (ENZYME CLASS)
EC 2.7.10.1
Created by admin on Tue Apr 01 23:42:39 GMT 2025 , Edited by admin on Tue Apr 01 23:42:39 GMT 2025
PRIMARY
From To
1_33 1_72
1_111 1_161
1_126 1_158
1_208 1_265
1_403 1_466
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_105
N 1_120
N 1_258
N 1_268
N 1_275
N 1_295
N 1_327
N 1_342
N 1_438
N 1_461
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR -> TARGET

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_796] [1_866] [1_934] DEXFOSFOSERINE VI4F0K069V
AMINO ACID SUBSTITUTION [1_716] [1_721] DEXFOSFOSERINE VI4F0K069V
AMINO ACID SUBSTITUTION [1_522] [1_528] [1_543] [1_545] [1_678] [1_696] [1_705] [1_798] [1_875] [1_911] TYROSINE O-PHOSPHATE 2R86C98KDX
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL