RU-24969 SUCCINATE

COc1ccc2c(c1)c(c[nH]2)C3=CCNCC3.C(CC(=O)O)C(=O)O

InChIKey=AFNQSRYIQUAMNM-UHFFFAOYSA-N

InChI=1S/C14H16N2O.C4H6O4/c1-17-11-2-3-14-12(8-11)13(9-16-14)10-4-6-15-7-5-10;5-3(6)1-2-4(7)8/h2-4,8-9,15-16H,5-7H2,1H3;1-2H2,(H,5,6)(H,7,8)

Stereochemistry	ACHIRAL
Additional Stereochemistry	No
Defined Stereocenters	0 / 0
E/Z Centers	0
Optical Activity	NONE

Stereochemistry	ACHIRAL
Additional Stereochemistry	No
Defined Stereocenters	0 / 0
E/Z Centers	0
Optical Activity	NONE

Targets

Primary Target	Pharmacology	Potency
Serotonin 6 (5-HT6) receptor 30 Target ID: CHEMBL3371 Sources: https://www.ncbi.nlm.nih.gov/pubmed/16055331	Agonist 2470	79.0 nM [IC50]
Serotonin 1a (5-HT1a) receptor 162 Target ID: CHEMBL214 Sources: https://www.ncbi.nlm.nih.gov/pubmed/9760039	Agonist 2470	1.13 nM [Ki]
Serotonin 1d (5-HT1d) receptor 46 Target ID: CHEMBL1983 Sources: https://www.ncbi.nlm.nih.gov/pubmed/1652050	Agonist 2470	18.0 nM [Ki]

Substance Class	Chemical Created by `admin` on `Sat Jun 26 16:33:06 UTC 2021` Edited by `admin` on `Sat Jun 26 16:33:06 UTC 2021`
Record UNII	RKG24J8KJR
Record Status	`Validated (UNII)`
Record Version

Name

Type

Language

RU-24969 SUCCINATE

Code

English

1H-INDOLE, 5-METHOXY-3-(1,2,3,6-TETRAHYDRO-4-PYRIDINYL)-, BUTANEDIOATE (1:1)

Systematic Name

English

Code System Code Type Description

CAS

107008-28-6

Created by admin on Sat Jun 26 16:33:07 UTC 2021 , Edited by admin on Sat Jun 26 16:33:07 UTC 2021

PRIMARY

PUBCHEM

108028

Created by admin on Sat Jun 26 16:33:07 UTC 2021 , Edited by admin on Sat Jun 26 16:33:07 UTC 2021

PRIMARY

FDA UNII

RKG24J8KJR

Created by admin on Sat Jun 26 16:33:07 UTC 2021 , Edited by admin on Sat Jun 26 16:33:07 UTC 2021

PRIMARY

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