U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 17:04:43 GMT 2025
Edited
by admin
on Tue Apr 01 17:04:43 GMT 2025
Protein Type ENZYME
Protein Sub Type TYROSINE KINASE
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
RGHTSAKWXW
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
CYTOPLASMIC TYROSINE-PROTEIN KINASE BMX
Common Name English
BONE MARROW TYROSINE KINASE GENE IN CHROMOSOME X PROTEIN
Preferred Name English
EPITHELIAL AND ENDOTHELIAL TYROSINE KINASE
Common Name English
NTK38
Common Name English
ETK
Common Name English
Code System Code Type Description
UNIPROT
P51813
Created by admin on Tue Apr 01 17:04:43 GMT 2025 , Edited by admin on Tue Apr 01 17:04:43 GMT 2025
PRIMARY
PHAROS
P51813
Created by admin on Tue Apr 01 17:04:43 GMT 2025 , Edited by admin on Tue Apr 01 17:04:43 GMT 2025
PRIMARY
FDA UNII
RGHTSAKWXW
Created by admin on Tue Apr 01 17:04:43 GMT 2025 , Edited by admin on Tue Apr 01 17:04:43 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_566] TYROSINE O-PHOSPHATE 2R86C98KDX
AMINO_ACID_SUBSTITUTION [1_121] [1_132] [1_133] [1_143] SITE_SPECIFIC C1H3-TYPE ZINC FINGER 0RK9393AEN
AMINO ACID SUBSTITUTION [1_216] [1_224] TYROSINE O-PHOSPHATE 2R86C98KDX
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL