Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 17:04:43 GMT 2025
by
admin
on
Tue Apr 01 17:04:43 GMT 2025
|
| Protein Type | ENZYME |
| Protein Sub Type | TYROSINE KINASE |
| Sequence Origin | HUMAN |
| Sequence Type | COMPLETE |
| Record UNII |
RGHTSAKWXW
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
|
Common Name | English | ||
|
Preferred Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
P51813
Created by
admin on Tue Apr 01 17:04:43 GMT 2025 , Edited by admin on Tue Apr 01 17:04:43 GMT 2025
|
PRIMARY | |||
|
P51813
Created by
admin on Tue Apr 01 17:04:43 GMT 2025 , Edited by admin on Tue Apr 01 17:04:43 GMT 2025
|
PRIMARY | |||
|
RGHTSAKWXW
Created by
admin on Tue Apr 01 17:04:43 GMT 2025 , Edited by admin on Tue Apr 01 17:04:43 GMT 2025
|
PRIMARY |
| Linkage Type | Residue Index | |||
|---|---|---|---|---|
| COORDINATION COMPOUND | 1_121 | 1_132 | 1_143 | 1_149 |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
IC50
|
Structural Modifications
| Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
|---|---|---|---|---|---|---|
| AMINO ACID SUBSTITUTION | [1_566] | TYROSINE O-PHOSPHATE | 2R86C98KDX | |||
| AMINO_ACID_SUBSTITUTION | [1_121] [1_132] [1_133] [1_143] | SITE_SPECIFIC | C1H3-TYPE ZINC FINGER | 0RK9393AEN | ||
| AMINO ACID SUBSTITUTION | [1_216] [1_224] | TYROSINE O-PHOSPHATE | 2R86C98KDX |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT | CHEMICAL |
|