U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Wed Apr 02 06:56:15 GMT 2025
Edited
by admin
on Wed Apr 02 06:56:15 GMT 2025
Protein Type ENZYME
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
QZ9EX1VZ9D
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
CYCLIN A2-CDK2 COMPLEX
Common Name English
CCNA2:CDK2 COMPLEX
Preferred Name English
CYCLIN-A2-CYCLIN-DEPENDENT KINASE 2 COMLEX
Common Name English
Code System Code Type Description
FDA UNII
QZ9EX1VZ9D
Created by admin on Wed Apr 02 06:56:15 GMT 2025 , Edited by admin on Wed Apr 02 06:56:15 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
Using the Nanosyn biochemical assay.
IC50
INHIBITOR -> TARGET

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO_ACID_SUBSTITUTION [2_6] SITE_SPECIFIC N6-ACETYLLYSINE 470AD5VY1X
AMINO_ACID_SUBSTITUTION [2_1] SITE_SPECIFIC N-ACETYLMETHIONINE 9J12WX5B6A
AMINO_ACID_SUBSTITUTION [2_14] [2_160] SITE_SPECIFIC THREONINE PHOSPHATE 3L4WX7B1EI
AMINO_ACID_SUBSTITUTION [2_15] [2_19] SITE_SPECIFIC TYROSINE O-PHOSPHATE 2R86C98KDX
AMINO_ACID_SUBSTITUTION [1_1] SITE_SPECIFIC N-ACETYLMETHIONINE 9J12WX5B6A
AMINO_ACID_SUBSTITUTION [1_5] [1_55] SITE_SPECIFIC DEXFOSFOSERINE VI4F0K069V
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL