U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Sat Dec 16 12:08:06 UTC 2023
Edited
by admin
on Sat Dec 16 12:08:06 UTC 2023
Protein Type RECEPTOR
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
QV1Q1KK8LA
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
MELANOCORTIN RECEPTOR 3
Common Name English
MC3-R
Common Name English
Code System Code Type Description
FDA UNII
QV1Q1KK8LA
Created by admin on Sat Dec 16 12:08:07 UTC 2023 , Edited by admin on Sat Dec 16 12:08:07 UTC 2023
PRIMARY
UNIPROT
P41968
Created by admin on Sat Dec 16 12:08:07 UTC 2023 , Edited by admin on Sat Dec 16 12:08:07 UTC 2023
PRIMARY
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_2
N 1_16
N 1_28
Related Record Type Details
INHIBITOR -> TARGET
BINDING
Ki
AGONIST -> TARGET
Ki
AGONIST -> TARGET
AGONIST -> TARGET
INHIBITOR -> TARGET
Ability to block α-MSH-induced cAMP production in a CHO cell line expressing hMC3R.
BIOASSAY (CELLULAR)
Ki
AGONIST -> TARGET
Biased agonist: AP1189 reduced cytokine release but no melanogenesis was induced.
AGONIST -> TARGET
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL