U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Wed Apr 02 02:40:32 GMT 2025
Edited
by admin
on Wed Apr 02 02:40:32 GMT 2025
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
Q8CNI6U44N
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
PSCTK4
Preferred Name English
TYROSINE-PROTEIN KINASE TEC
Common Name English
TEC
Common Name English
Code System Code Type Description
PHAROS
P42680
Created by admin on Wed Apr 02 02:40:32 GMT 2025 , Edited by admin on Wed Apr 02 02:40:32 GMT 2025
PRIMARY
WIKIPEDIA
TRPV1
Created by admin on Wed Apr 02 02:40:32 GMT 2025 , Edited by admin on Wed Apr 02 02:40:32 GMT 2025
PRIMARY
FDA UNII
Q8CNI6U44N
Created by admin on Wed Apr 02 02:40:32 GMT 2025 , Edited by admin on Wed Apr 02 02:40:32 GMT 2025
PRIMARY
UNIPROT
P42680
Created by admin on Wed Apr 02 02:40:32 GMT 2025 , Edited by admin on Wed Apr 02 02:40:32 GMT 2025
PRIMARY
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_253
N 1_538
Related Record Type Details
INHIBITOR -> TARGET
77.6 % inhibition at 1 micromolar
IC50
INHIBITOR -> TARGET

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_228] TYROSINE O-PHOSPHATE 2R86C98KDX
Name Property Type Amount Referenced Substance Defining Parameters References
Molecular Formula CHEMICAL
MOL_WEIGHT CHEMICAL