Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 19:39:48 GMT 2025
by
admin
on
Tue Apr 01 19:39:48 GMT 2025
|
| Protein Sub Type | |
| Sequence Type | COMPLETE |
| Record UNII |
Q43F7CTH27
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
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Preferred Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
|
Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
Q9GZT9
Created by
admin on Tue Apr 01 19:39:48 GMT 2025 , Edited by admin on Tue Apr 01 19:39:48 GMT 2025
|
PRIMARY | |||
|
Q9GZT9
Created by
admin on Tue Apr 01 19:39:48 GMT 2025 , Edited by admin on Tue Apr 01 19:39:48 GMT 2025
|
PRIMARY | |||
|
EGLN1
Created by
admin on Tue Apr 01 19:39:48 GMT 2025 , Edited by admin on Tue Apr 01 19:39:48 GMT 2025
|
PRIMARY | |||
|
Q43F7CTH27
Created by
admin on Tue Apr 01 19:39:48 GMT 2025 , Edited by admin on Tue Apr 01 19:39:48 GMT 2025
|
PRIMARY |
| Linkage Type | Residue Index | |||
|---|---|---|---|---|
| COORDINATION COMPOUND | 1_312 | 1_314 | 1_373 | |
| COORDINATION COMPOUND | 1_20 | 1_23 | 1_32 | 1_35 |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
INHIBITOR -> TARGET |
|
||
|
INHIBITOR -> TARGET |
Ki
|
||
|
INHIBITOR -> TARGET |
PRECLINICAL
|
||
|
|
INHIBITOR -> TARGET |
IC50
|
Structural Modifications
| Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
|---|---|---|---|---|---|---|
| AMINO_ACID_SUBSTITUTION | [1_312] [1_314] [1_373] | SITE_SPECIFIC | PROLYL HYDROXYLASE IRON BINDING SITE | 6W7112Q7X7 | ||
| AMINO ACID SUBSTITUTION | [1_200] [1_207] [1_301] [1_322] [1_325] | S-NITROSOCYSTEINE | 926P2322P4 | |||
| AMINO_ACID_SUBSTITUTION | [1_20] [1_23] [1_32] [1_35] | SITE_SPECIFIC | C4-TYPE ZINC FINGER | C56TF4V7OP |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT | CHEMICAL |
|