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Details

Stereochemistry ABSOLUTE
Molecular Formula C46H58N4O10
Molecular Weight 826.9735
Optical Activity UNSPECIFIED
Defined Stereocenters 10 / 10
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of Vinblastine N-Oxide

SMILES

CC[C@]1(O)C[C@@H]2C[N@+]([O-])(C1)CCC3=C(NC4=C3C=CC=C4)[C@@](C2)(C(=O)OC)C5=C(OC)C=C6N(C)[C@@H]7[C@]8(CCN9CC=C[C@](CC)([C@@H]89)[C@@H](OC(C)=O)[C@]7(O)C(=O)OC)C6=C5

InChI

InChIKey=JJNRGDILJOBAEK-FFFVJEPASA-N
InChI=1S/C46H58N4O10/c1-8-42(54)23-28-24-45(40(52)58-6,36-30(15-20-50(56,25-28)26-42)29-13-10-11-14-33(29)47-36)32-21-31-34(22-35(32)57-5)48(4)38-44(31)17-19-49-18-12-16-43(9-2,37(44)49)39(60-27(3)51)46(38,55)41(53)59-7/h10-14,16,21-22,28,37-39,47,54-55H,8-9,15,17-20,23-26H2,1-7H3/t28-,37-,38+,39+,42-,43+,44+,45-,46-,50-/m0/s1

HIDE SMILES / InChI

Molecular Formula C46H58N4O10
Molecular Weight 826.9735
Charge 0
Count
Stereochemistry ABSOLUTE
Additional Stereochemistry No
Defined Stereocenters 10 / 10
E/Z Centers 0
Optical Activity UNSPECIFIED

Approval Year

Substance Class Chemical
Created
by admin
on Wed Apr 02 14:08:09 GMT 2025
Edited
by admin
on Wed Apr 02 14:08:09 GMT 2025
Record UNII
PN45E4NV2N
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
CPD-100
Preferred Name English
Vinblastine N-Oxide
Common Name English
Vinblastine N'b-oxide
Common Name English
Vincaleukoblastine, 6?-oxide
Common Name English
Vinblastine Impurity B
Common Name English
Classification Tree Code System Code
FDA ORPHAN DRUG 904922
Created by admin on Wed Apr 02 14:08:09 GMT 2025 , Edited by admin on Wed Apr 02 14:08:09 GMT 2025
Code System Code Type Description
CAS
61936-68-3
Created by admin on Wed Apr 02 14:08:09 GMT 2025 , Edited by admin on Wed Apr 02 14:08:09 GMT 2025
PRIMARY
PUBCHEM
166177221
Created by admin on Wed Apr 02 14:08:09 GMT 2025 , Edited by admin on Wed Apr 02 14:08:09 GMT 2025
PRIMARY
FDA UNII
PN45E4NV2N
Created by admin on Wed Apr 02 14:08:09 GMT 2025 , Edited by admin on Wed Apr 02 14:08:09 GMT 2025
PRIMARY
Related Record Type Details
METABOLITE ACTIVE -> PRODRUG
Name Property Type Amount Referenced Substance Defining Parameters References
Route of Elimination PHARMACOKINETIC
Biological Half-life PHARMACOKINETIC
Route of Elimination PHARMACOKINETIC