Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Sat Dec 16 14:58:39 GMT 2023
by
admin
on
Sat Dec 16 14:58:39 GMT 2023
|
| Protein Sub Type | |
| Sequence Type | COMPLETE |
| Record UNII |
PIV978KC1N
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
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P35498
Created by
admin on Sat Dec 16 14:58:40 GMT 2023 , Edited by admin on Sat Dec 16 14:58:40 GMT 2023
|
PRIMARY | |||
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PIV978KC1N
Created by
admin on Sat Dec 16 14:58:40 GMT 2023 , Edited by admin on Sat Dec 16 14:58:40 GMT 2023
|
PRIMARY |
| Glycosylation Type | HUMAN |
| Glycosylation Link Type | Site |
|---|---|
| N | 1_211 |
| N | 1_284 |
| N | 1_295 |
| N | 1_301 |
| N | 1_306 |
| N | 1_338 |
| N | 1_1378 |
| N | 1_1392 |
| N | 1_1403 |
| Related Record | Type | Details | ||
|---|---|---|---|---|
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
Shifts hNav1.1 opening to more depolarized voltages without further alterations in the gating properties of hNav1.1, hNav1.2, hNav1.3, and hNav1.6;
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
Binds to inactivated state and prevents activation
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
EC50
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INDUCER OF EXPRESSION->TARGET |
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| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT | CHEMICAL |
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| Molecular Formula | CHEMICAL |
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