B1 BRADYKININ RECEPTOR

Approval Year

Substance Class	Protein Created by `admin` on `Tue Apr 01 17:32:15 GMT 2025` Edited by `admin` on `Tue Apr 01 17:32:15 GMT 2025`
Protein Type	RECEPTOR
Protein Sub Type
Sequence Origin	HUMAN
Sequence Type	COMPLETE
Record UNII	PI5P4K0HAG
Record Status	`Validated (UNII)`
Record Version

Download

Name

Type

Language

B1 BRADYKININ RECEPTOR

Common Name

English

B1R

Preferred Name

English

BK-1 RECEPTOR

Common Name

English

BRADYB1

Common Name

English

Code System Code Type Description

FDA UNII

PI5P4K0HAG

Created by admin on Tue Apr 01 17:32:15 GMT 2025 , Edited by admin on Tue Apr 01 17:32:15 GMT 2025

PRIMARY

UNIPROT

P46663

Created by admin on Tue Apr 01 17:32:15 GMT 2025 , Edited by admin on Tue Apr 01 17:32:15 GMT 2025

PRIMARY

From	To
1_110	1_189

Glycosylation Type

HUMAN

Glycosylation Link Type	Site
N	1_14
N	1_22
N	1_185

Related Record Type Details


					58QE2VVE3Q

DABK

AGONIST -> TARGET

Amount:


					Z93D4NV99S

Fulimetibant

INHIBITOR -> TARGET

Interaction Type:

PRECLINICAL

Amount:


					02HU8HWP7U

SAFOTIBANT

INHIBITOR -> TARGET

Qualification:

Ki

Amount:


					189R4J5E0F

SSR-240612 FREE BASE

INHIBITOR -> TARGET

Comments:

Functional assay measuring inhibition of inositol phosphate-1 formation induced by Lys0-desArg9- BK in activation of the B1 receptor in MRC5 human fibroblast cells.

Qualification:

IC50

Amount: