U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Sat Dec 16 11:38:52 GMT 2023
Edited
by admin
on Sat Dec 16 11:38:52 GMT 2023
Protein Sub Type
Sequence Type COMPLETE
Record UNII
PG244BS39U
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
BETA-3 ADRENERGIC RECEPTOR
Common Name English
B3AR
Common Name English
ADRB3R
Common Name English
beta3
Common Name English
β3-Adrenergic Receptor
Common Name English
Code System Code Type Description
FDA UNII
PG244BS39U
Created by admin on Sat Dec 16 11:38:53 GMT 2023 , Edited by admin on Sat Dec 16 11:38:53 GMT 2023
PRIMARY
PHAROS
P13945
Created by admin on Sat Dec 16 11:38:53 GMT 2023 , Edited by admin on Sat Dec 16 11:38:53 GMT 2023
PRIMARY
WIKIPEDIA
BETA-3_ADRENERGIC_RECEPTOR
Created by admin on Sat Dec 16 11:38:53 GMT 2023 , Edited by admin on Sat Dec 16 11:38:53 GMT 2023
PRIMARY
UNIPROT
P13945
Created by admin on Sat Dec 16 11:38:53 GMT 2023 , Edited by admin on Sat Dec 16 11:38:53 GMT 2023
PRIMARY
From To
1_110 1_196
1_189 1_195
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_8
N 1_26
Related Record Type Details
INHIBITOR -> TARGET
AGONIST -> TARGET
EC50
RADIOLIGAND->TARGET
Chinese hamster ovary (CHO) cells stably expressing the three β-adrenergic receptor subtypes at comparable levels.
Kd
TARGET->WEAK AGONIST
Assay in chinese hamster ovary (CHO) cells stably expressing the three β-adrenergic receptor subtypes at comparable leve50 to 80 pM 125I-CYP were used as radioligand. Experiments were done in the presence of 100 µM GTP.
Ki
INHIBITOR -> TARGET
Chinese hamster ovary (CHO) cells stably expressing the three β-adrenergic receptor subtypes at comparable levels.
Kd
AGONIST -> TARGET
SHORT-ACTING
AGONIST -> TARGET
Assay in chinese hamster ovary (CHO) cells stably expressing the three β-adrenergic receptor subtypes at comparable leve50 to 80 pM 125I-CYP were used as radioligand. Experiments were done in the presence of 100 µM GTP.
Ki
AGONIST -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
SELECTIVE
AGONIST -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
SHORT-ACTING
AGONIST -> TARGET
AGONIST -> TARGET
SHORT-ACTING
AGONIST -> TARGET
SHORT-ACTING
AGONIST -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
Assay in chinese hamster ovary (CHO) cells stably expressing the three β-adrenergic receptor subtypes at comparable leve50 to 80 pM 125I-CYP were used as radioligand. Experiments were done in the presence of 100 µM GTP.
AGONIST -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
SHORT-ACTING
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL
Molecular Formula CHEMICAL