U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 18:22:09 GMT 2025
Edited
by admin
on Tue Apr 01 18:22:09 GMT 2025
Protein Sub Type
Sequence Type COMPLETE
Record UNII
OUJ3871L27
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
GASTRIN-RELEASING PEPTIDE RECEPTOR
Common Name English
GRP-PREFERRING BOMBESIN RECEPTOR
Preferred Name English
GRP-R
Common Name English
Code System Code Type Description
FDA UNII
OUJ3871L27
Created by admin on Tue Apr 01 18:22:09 GMT 2025 , Edited by admin on Tue Apr 01 18:22:09 GMT 2025
PRIMARY
From To
1_113 1_196
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_20
Related Record Type Details
RADIOLIGAND->TARGET
Expression in prostate cancer is higher in carcinomas of lower Gleason score. GRP-R imaging appears complimentary to that of imaging prostate-specific membrane antigen.
Kd
RADIOLIGAND->TARGET
RADIOLIGAND->TARGET
INHIBITOR -> TARGET
Pre-clinical
LIGAND->TARGET
INHIBITOR -> TARGET
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL