U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS
This repository is under review for potential modification in compliance with Administration directives.

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 17:29:58 GMT 2025
Edited
by admin
on Tue Apr 01 17:29:58 GMT 2025
Protein Sub Type
Sequence Type COMPLETE
Record UNII
OD27Q24FJ4
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
ARK-1
Preferred Name English
AURORA KINASE A
Common Name English
SERINE/THREONINE-PROTEIN KINASE 15
Common Name English
AURKA
Common Name English
SERINE/THREONINE-PROTEIN KINASE AURORA-A
Common Name English
AURORA 2
Common Name English
AURORA/IPL1-RELATED KINASE 1
Common Name English
SERINE/THREONINE-PROTEIN KINASE 6
Common Name English
AURORA-RELATED KINASE 1
Common Name English
Code System Code Type Description
PHAROS
O14965
Created by admin on Tue Apr 01 17:29:58 GMT 2025 , Edited by admin on Tue Apr 01 17:29:58 GMT 2025
PRIMARY
FDA UNII
OD27Q24FJ4
Created by admin on Tue Apr 01 17:29:58 GMT 2025 , Edited by admin on Tue Apr 01 17:29:58 GMT 2025
PRIMARY
UNIPROT
O14965
Created by admin on Tue Apr 01 17:29:58 GMT 2025 , Edited by admin on Tue Apr 01 17:29:58 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR->OFF-TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
COMPETITIVE INHIBITOR
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
COMPETITIVE INHIBITOR
IC50

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_287] [1_288] THREONINE PHOSPHATE 3L4WX7B1EI
AMINO ACID SUBSTITUTION [1_41] [1_51] DEXFOSFOSERINE VI4F0K069V
AMINO ACID SUBSTITUTION [1_342] DEXFOSFOSERINE VI4F0K069V
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL