U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS
This repository is under review for potential modification in compliance with Administration directives.

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 18:32:35 GMT 2025
Edited
by admin
on Tue Apr 01 18:32:35 GMT 2025
Protein Sub Type
Sequence Type COMPLETE
Record UNII
O0QUP6NQ1H
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
P2Y PURINOCEPTOR 12
Common Name English
ADP-GLUCOSE RECEPTOR
Preferred Name English
P2Y12
Common Name English
SP1999
Common Name English
ADPG-R
Common Name English
P2Y(CYC)
Common Name English
HORK3
Common Name English
P2Y(AC)
Common Name English
P2Y12 PLATELET ADP RECEPTOR
Common Name English
Code System Code Type Description
UNIPROT
Q9H244
Created by admin on Tue Apr 01 18:32:35 GMT 2025 , Edited by admin on Tue Apr 01 18:32:35 GMT 2025
PRIMARY
FDA UNII
O0QUP6NQ1H
Created by admin on Tue Apr 01 18:32:35 GMT 2025 , Edited by admin on Tue Apr 01 18:32:35 GMT 2025
PRIMARY
PHAROS
Q9H244
Created by admin on Tue Apr 01 18:32:35 GMT 2025 , Edited by admin on Tue Apr 01 18:32:35 GMT 2025
PRIMARY
From To
1_17 1_270
1_97 1_175
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_6
N 1_13
Related Record Type Details
AGONIST -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IN-VITRO
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
AGONIST -> TARGET
Leads to platelet activation
INHIBITOR -> TARGET
INHIBITOR -> TARGET

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_55] [1_57] DEXFOSFOSERINE VI4F0K069V
Name Property Type Amount Referenced Substance Defining Parameters References
Molecular Formula CHEMICAL
MOL_WEIGHT CHEMICAL